SCHEMBL21744950

SCHEMBL21744950

CC(O)c1ccc(-n2cccn2)nc1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.54
KMT2A Q03164 2/20 0.52
KDM4E B2RXH2 6/20 0.47
ALDH1A1 P00352 2/20 0.46
RXFP1 Q9HBX9 1/20 0.46
OGA O60502 1/20 0.45
MEN1 O00255 1/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP2D6 P10635 1/20 0.43
KDM5B Q9UGL1 1/20 0.41
HPGD P15428 2/20 0.41
TNIK Q9UKE5 1/20 0.41
GRN P28799 1/20 0.40
SORT1 Q99523 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
CHRNA7 P36544 1/20 0.40
PCSK9 Q8NBP7 1/20 0.39
CXCR4 P61073 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12680212 0.87 LMNA (0.53) LMNAKMT2AKDM4EALDH1A1RXFP1
SCHEMBL25560876 0.84 LMNA (0.50) LMNAKMT2AKDM4EALDH1A1RXFP1
SCHEMBL23957682 0.82 LMNA (0.48) LMNAKMT2AKDM4EALDH1A1RXFP1
SCHEMBL20372859 0.82 LMNA (0.48) LMNAKMT2AKDM4EALDH1A1RXFP1
SCHEMBL28938107 0.78 LMNA (0.51) LMNAKMT2AKDM4EALDH1A1RXFP1
SCHEMBL23352193 0.76 LMNA (0.45) LMNAKMT2AKDM4EALDH1A1RXFP1
SCHEMBL24724171 0.75 KDM4E (0.44) LMNAKMT2AKDM4EALDH1A1OGA
SCHEMBL31516755 0.75 KDM4E (0.58) LMNAKMT2AKDM4EALDH1A1RXFP1
SCHEMBL861501 0.75 LMNA (0.61) LMNAKMT2AKDM4EALDH1A1RXFP1
SCHEMBL46317 0.75 KDM4E (0.58) LMNAKMT2AKDM4EALDH1A1RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020035065-A1 PYRAZOLE DERIVATIVE AS RET INHIBITOR 南京明德新药研发有限公司 2020-02-20 WO disclosed