SCHEMBL21751708

SCHEMBL21751708

C[Si](C)(C)CCOCn1ccc2cc(Br)c(O)nc21

nearest known ligand 0.38

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 3/20 0.38
NPC1 O15118 1/20 0.33
KLKB1 P03952 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19203911 0.86 DGAT1 (0.41) DGAT1NPC1KLKB1
SCHEMBL20553711 0.85 DGAT1 (0.37) DGAT1NPC1KLKB1
SCHEMBL21751697 0.85 DGAT1 (0.38) DGAT1NPC1
SCHEMBL20767635 0.85 NPC1 (0.35) DGAT1NPC1KLKB1
SCHEMBL30074962 0.85 DGAT1 (0.38) DGAT1NPC1
SCHEMBL20767549 0.85 DGAT1 (0.46) DGAT1NPC1
SCHEMBL25349464 0.84 DGAT1 (0.38) DGAT1NPC1
Hydrochloric Acid SCHEMBL29722941 0.84 NPC1 (0.34) DGAT1NPC1KLKB1
Hydrochloric Acid SCHEMBL20767619 0.84 NPC1 (0.34) DGAT1NPC1KLKB1
Hydrochloric Acid SCHEMBL20767618 0.82 NPC1 (0.34) DGAT1NPC1KLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12220419-B2 BCL-2 inhibitors NEWAVE PHARMACEUTICAL INC. (US) 2025-02-11 US disclosed
US-20230295183-A1 HOT MELT EXTRUDED SOLID DISPERSIONS CONTAINING A BCL2 INHIBITOR NEWAVE PHARMACEUTICAL INC. 2023-09-21 US disclosed
CN-116270660-A Bcl-2/Bcl-xl inhibitor-containing composition and preparation method and application thereof 广州麓鹏制药有限公司 2023-06-23 CN disclosed
CN-116236583-A Bcl-2/Bcl-xl inhibitor-containing composition and preparation method and application thereof 广州麓鹏制药有限公司 2023-06-09 CN disclosed
EP-4110298-A1 HOT MELT EXTRUDED SOLID DISPERSIONS CONTAINING A BCL2 INHIBITOR Guangzhou Lupeng Pharmaceutical Company Ltd. (CN) 2023-01-04 EP disclosed
CN-115484933-A Hot melt extrusion solid dispersions containing BCL2 inhibitors 广州麓鹏制药有限公司 2022-12-16 CN disclosed
US-20220372042-A1 CONDENSED HETEROCYCLES AS BCL-2 INHIBITORS NEWAVE PHARMACEUTICAL INC. 2022-11-24 US disclosed
US-20210315904-A1 BCL-2 INHIBITORS NEWAVE PHARMACEUTICAL INC. 2021-10-14 US disclosed
WO-2021066873-A1 CONDENSED HETEROCYCLES AS BCL-2 INHIBITORS NEWAVE PHARMACEUTICAL INC. (US) 2021-04-08 WO disclosed
WO-2020041406-A1 BCL-2 INHIBITORS NEWAVE PHARMACEUTICAL INC. (US) 2020-02-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230295183-A1 HOT MELT EXTRUDED SOLID DISPERSIONS CONTAINING A BCL2 INHIBITOR BCL2, BCL2L1, BCL2L2 DGAT1 3779/4885NPC1 2558/4885KLKB1 3509/4885
US-20210315904-A1 BCL-2 INHIBITORS BCL2L10, BCL2, BCL2L11 DGAT1 4227/4885NPC1 3788/4885KLKB1 3570/4885
US-12220419-B2 BCL-2 inhibitors BCL2L10, BCL2, BCL2L11 DGAT1 4227/4885NPC1 3788/4885KLKB1 3570/4885
US-20220372042-A1 CONDENSED HETEROCYCLES AS BCL-2 INHIBITORS BCL2L11, BCL2L10, BCL2 DGAT1 4510/4885NPC1 3924/4885KLKB1 2992/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.