SCHEMBL21752896

SCHEMBL21752896

CSc1cc(F)cc(C2CC(F)CN2c2ccc3ncc(C(=O)NC4CCN(Cc5ccc(F)c(O)c5)CC4)n3n2)c1

nearest known ligand 0.37

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 12/20 0.37
CCR3 P51677 5/20 0.35
MCHR1 Q99705 4/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21752901 1.00 NTRK1 (0.37) NTRK1CCR3MCHR1
SCHEMBL30032192 1.00 NTRK1 (0.37) NTRK1CCR3MCHR1
SCHEMBL30033137 1.00 NTRK1 (0.37) NTRK1CCR3MCHR1
SCHEMBL30033807 0.97 CCR3 (0.37) NTRK1CCR3MCHR1
SCHEMBL30032907 0.97 CCR3 (0.37) NTRK1CCR3MCHR1
SCHEMBL21752874 0.97 CCR3 (0.37) NTRK1CCR3MCHR1
SCHEMBL21752813 0.97 CCR3 (0.37) NTRK1CCR3MCHR1
SCHEMBL21752906 0.94 NTRK1 (0.35) NTRK1
SCHEMBL21752905 0.94 NTRK1 (0.35) NTRK1
SCHEMBL21752927 0.91 NTRK1 (0.41) NTRK1CCR3MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112805062-B Imidazo [1,2-b ] pyridazines as Trk inhibitors 博善人工智能生物科技有限公司 2024-06-04 CN claimed
EP-3840832-B1 IMIDAZO[1,2-B]PYRIDAZINES AS TRK INHIBITORS BENEVOLENTAI BIO LTD (GB) 2023-10-11 EP claimed
US-20230149398-A1 TOPICAL PHARMACEUTICAL COMPOSITIONS COMPRISING IMIDAZO[1,2-B]PYRIDAZINE COMPOUNDS BENEVOLENTAI BIO LIMITED (GB) 2023-05-18 US claimed
EP-4093404-A1 TOPICAL PHARMACEUTICAL COMPOSITIONS COMPRISING IMIDAZO[1,2-B]PYRIDAZINE COMPOUNDS BenevolentAI Bio Limited (GB) 2022-11-30 EP claimed
CN-115297863-A Topical pharmaceutical compositions comprising imidazo [1,2-b ] pyridazine compounds 博善人工智能生物科技有限公司 2022-11-04 CN claimed
US-20210253572-A1 IMIDAZO[1,2-B]PYRIDAZINES AS TRK INHIBITORS BenevolentAl Bio Limited (GB) 2021-08-19 US claimed
WO-2021148805-A1 TOPICAL PHARMACEUTICAL COMPOSITIONS COMPRISING IMIDAZO[1,2-B]PYRIDAZINE COMPOUNDS BENEVOLENTAI BIO LIMITED (GB) 2021-07-29 WO claimed
EP-3840832-A1 IMIDAZO[1,2-B]PYRIDAZINES AS TRK INHIBITORS BenevolentAI Bio Limited (GB) 2021-06-30 EP claimed
CN-112805062-A Imidazo [1,2-b ] pyridazines as Trk inhibitors 博善人工智能生物科技有限公司 2021-05-14 CN claimed
WO-2020039209-A1 IMIDAZO[1,2-B]PYRIDAZINES AS TRK INHIBITORS BENEVOLENTAI BIO LIMITED (GB) 2020-02-27 WO claimed
CN-112805062-B Imidazo [1,2-b ] pyridazines as Trk inhibitors 博善人工智能生物科技有限公司 2024-06-04 CN disclosed
EP-3840832-B1 IMIDAZO[1,2-B]PYRIDAZINES AS TRK INHIBITORS BENEVOLENTAI BIO LTD (GB) 2023-10-11 EP disclosed
US-20230149398-A1 TOPICAL PHARMACEUTICAL COMPOSITIONS COMPRISING IMIDAZO[1,2-B]PYRIDAZINE COMPOUNDS BENEVOLENTAI BIO LIMITED (GB) 2023-05-18 US disclosed
EP-4093404-A1 TOPICAL PHARMACEUTICAL COMPOSITIONS COMPRISING IMIDAZO[1,2-B]PYRIDAZINE COMPOUNDS BenevolentAI Bio Limited (GB) 2022-11-30 EP disclosed
CN-115297863-A Topical pharmaceutical compositions comprising imidazo [1,2-b ] pyridazine compounds 博善人工智能生物科技有限公司 2022-11-04 CN disclosed
US-20210253572-A1 IMIDAZO[1,2-B]PYRIDAZINES AS TRK INHIBITORS BenevolentAl Bio Limited (GB) 2021-08-19 US disclosed
WO-2021148805-A1 TOPICAL PHARMACEUTICAL COMPOSITIONS COMPRISING IMIDAZO[1,2-B]PYRIDAZINE COMPOUNDS BENEVOLENTAI BIO LIMITED (GB) 2021-07-29 WO disclosed
EP-3840832-A1 IMIDAZO[1,2-B]PYRIDAZINES AS TRK INHIBITORS BenevolentAI Bio Limited (GB) 2021-06-30 EP disclosed
CN-112805062-A Imidazo [1,2-b ] pyridazines as Trk inhibitors 博善人工智能生物科技有限公司 2021-05-14 CN disclosed
WO-2020039209-A1 IMIDAZO[1,2-B]PYRIDAZINES AS TRK INHIBITORS BENEVOLENTAI BIO LIMITED (GB) 2020-02-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230149398-A1 TOPICAL PHARMACEUTICAL COMPOSITIONS COMPRISING IMIDAZO[1,2-B]PYRIDAZINE COMPOUNDS TNK2, TNIK, TNK1 NTRK1 15/4885CCR3 2473/4885MCHR1 3603/4885
US-20210253572-A1 IMIDAZO[1,2-B]PYRIDAZINES AS TRK INHIBITORS MUSK, TPM3, CSNK1A1 NTRK1 6/4885CCR3 3320/4885MCHR1 3842/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.