SCHEMBL21753834

SCHEMBL21753834

CC(N)CCCC(C)(C)N

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.46
ALDH1A1 P00352 3/20 0.43
TDP1 Q9NUW8 1/20 0.43
TP53 P04637 1/20 0.41
GABRP O00591 2/20 0.37
GABRD O14764 2/20 0.37
GABRA1 P14867 2/20 0.37
GABRB1 P18505 2/20 0.37
GABRG2 P18507 2/20 0.37
GABRB3 P28472 2/20 0.37
GABRA5 P31644 2/20 0.37
GABRA3 P34903 2/20 0.37
GABRA2 P47869 2/20 0.37
GABRB2 P47870 2/20 0.37
GABRA4 P48169 2/20 0.37
GABRE P78334 2/20 0.37
GABRA6 Q16445 2/20 0.37
GABRG1 Q8N1C3 2/20 0.37
GABRG3 Q99928 2/20 0.37
GABRQ Q9UN88 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3886965 0.83
SCHEMBL29240935 0.81 OPRM1 (0.34) OPRM1ALDH1A1
SCHEMBL3655016 0.81 OPRM1 (0.48) OPRM1ALDH1A1TDP1TP53GABRP
SCHEMBL4692345 0.81 CYP3A4 (0.42) ALDH1A1GRM4
Hydrochloric Acid SCHEMBL5463903 0.81 OPRM1 (0.36) OPRM1ALDH1A1TDP1GABRPGABRD
SCHEMBL28732357 0.80 OPRM1 (0.42) OPRM1ALDH1A1TDP1TP53GABRP
SCHEMBL11381711 0.80 TRPV1 (0.36) GRM4TRPV1TRPA1
Heptaminol SCHEMBL7530730 0.79 OPRM1 (0.46) OPRM1ALDH1A1TDP1TP53GABRP
Heptaminol SCHEMBL3163491 0.79 OPRM1 (0.46) OPRM1ALDH1A1TDP1TP53GABRP
Heptaminol SCHEMBL152610 0.79 OPRM1 (0.46) OPRM1ALDH1A1TDP1TP53GABRP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118344372-A Substituted straight-chain spiro derivatives 詹森药业有限公司 2024-07-16 CN disclosed
CN-118255774-A Substituted straight-chain spiro derivatives 詹森药业有限公司 2024-06-28 CN disclosed
CN-118255773-A Substituted straight-chain spiro derivatives 詹森药业有限公司 2024-06-28 CN disclosed
CN-117597348-A (R) -N-ethyl-5-fluoro-N-isopropyl-2- ((5- (2- (6- ((2-methoxyethyl) (methyl) amino) -2-methylhex-3-yl) -2, 6-diazaspiro [3.4] oct-6-yl) -1,2, 4-triazin-6-yl) oxy) benzamide benzenesulfonate for the treatment of diseases such as cancer 詹森药业有限公司 2024-02-23 CN disclosed
CN-117460513-A Combination therapy 詹森药业有限公司 2024-01-26 CN disclosed
CN-117337180-A combination therapy 詹森药业有限公司 2024-01-02 CN disclosed
CN-110770271-B Method for preparing functionalized fluorinated monomers, fluorinated monomers and compositions for preparing same 埃特纳科技有限公司 2023-04-18 CN disclosed
CN-114867721-A Substituted straight-chain spiro derivatives 詹森药业有限公司 2022-08-05 CN disclosed
WO-2020040283-A1 POLYAMIDE COMPOSITION 株式会社クラレ 2020-02-27 WO disclosed
WO-2020040282-A1 POLYAMIDE AND POLYAMIDE COMPOSITION 株式会社クラレ 2020-02-27 WO disclosed
CN-101180322-A Process for producing aqueous polymer dispersions BASF AG (DE) 2008-05-14 CN disclosed