SCHEMBL21753969

SCHEMBL21753969

COCOc1cc(N)c(C(C)=O)cc1OC

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.54
HTT P42858 3/20 0.49
CYP3A4 P08684 3/20 0.44
TSHR P16473 1/20 0.44
GAA P10253 1/20 0.39
HMGCR P04035 1/20 0.38
LMNA P02545 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.37
RAB9A P51151 1/20 0.37
LCK P06239 1/20 0.37
FYN P06241 1/20 0.37
POLB P06746 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30870738 0.87 KDM4E (0.69) KDM4EHTTCYP3A4TSHRGAA
SCHEMBL705665 0.87 KDM4E (0.69) KDM4EHTTCYP3A4TSHRGAA
SCHEMBL4770365 0.86 KDM4E (0.53) KDM4EHTTCYP3A4TSHRGAA
SCHEMBL6096678 0.86 KDM4E (0.53) KDM4EHTTCYP3A4TSHRGAA
SCHEMBL7300064 0.86 TSHR (0.62) KDM4EHTTCYP3A4TSHRGAA
SCHEMBL7291805 0.86 TSHR (0.62) KDM4EHTTCYP3A4TSHRGAA
SCHEMBL16285129 0.84 KDM4E (0.54) KDM4EHTTCYP3A4TSHRGAA
SCHEMBL19364180 0.83 CYP3A4 (0.58) KDM4EHTTCYP3A4TSHRHMGCR
SCHEMBL16280043 0.82 KDM4E (0.51) KDM4EHTTCYP3A4TSHRGAA
SCHEMBL16083519 0.82 KDM4E (0.51) KDM4EHTTCYP3A4TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020040581-A1 NOVEL QUINOLINE DERIVATIVE OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, AND PHARMACEUTICAL COMPOSITION CONTAINING SAME AS ACTIVE INGREDIENT 고려대학교 산학협력단 2020-02-27 WO disclosed