SCHEMBL705665

SCHEMBL705665

COc1cc(N)c(C(C)=O)cc1OC

nearest known ligand 0.69

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.69
HTT P42858 2/20 0.62
CYP3A4 P08684 3/20 0.52
GAA P10253 1/20 0.47
LCK P06239 1/20 0.46
FYN P06241 1/20 0.46
POLB P06746 1/20 0.44
LMNA P02545 2/20 0.44
ALDH1A1 P00352 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
RAB9A P51151 1/20 0.44
HMGCR P04035 1/20 0.43
KMT2A Q03164 1/20 0.42
PDE4A P27815 1/20 0.41
TNFSF11 O14788 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30870738 1.00 KDM4E (0.69) KDM4EHTTCYP3A4GAALCK
SCHEMBL26027709 0.90 KDM4E (0.56) KDM4EHTTCYP3A4GAALCK
SCHEMBL7300064 0.88 TSHR (0.62) KDM4EHTTCYP3A4GAARAB9A
SCHEMBL7291805 0.88 TSHR (0.62) KDM4EHTTCYP3A4GAARAB9A
SCHEMBL16285129 0.87 KDM4E (0.54) KDM4EHTTCYP3A4GAALCK
SCHEMBL21753969 0.87 KDM4E (0.54) KDM4EHTTCYP3A4GAALCK
SCHEMBL12793494 0.86 HTT (0.56) KDM4EHTTCYP3A4GAALMNA
SCHEMBL10520470 0.86 KDM4E (0.53) KDM4EHTTCYP3A4GAAPOLB
SCHEMBL4770365 0.85 KDM4E (0.53) KDM4EHTTCYP3A4GAAPOLB
SCHEMBL6096678 0.85 KDM4E (0.53) KDM4EHTTCYP3A4GAAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 264 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102532116-B Synthesis method of anti-tumor targeted therapeutic drug tivozanib WUHAN MAIDESEN MEDICAL TECHNOLOGY CO LTD 2015-01-21 CN claimed
EP-1506196-B1 PYRAZOLOPYRIMIDINES AS SODIUM CHANNEL INHIBITORS ICAGEN INC (US) 2012-01-18 EP claimed
US-5672352-A Methods of identifying the avian repellent effects of a compound and methods of repelling birds from materials susceptible to consumption by birds MONELL CHEMICAL SENSES CENTER (US) 1997-09-30 US claimed
US-20260022135-A1 ECTONUCLEOTIDE PYROPHOSPHATASE-PHOSPHODIESTERASE-1 (ENPP1) INHIBITORS AND USES THEREOF 1CBIO INC (US) 2026-01-22 US disclosed
US-12325720-B2 Ectonucleotide pyrophosphatase-phosphodiesterase-1 (ENPP1) inhibitors and uses thereof 1CBIO, INC. (US) 2025-06-10 US disclosed
WO-2025062157-A1 NEW TREATMENTS FOR PAIN SEVENLESS THERAPEUTICS LIMITED (GB) 2025-03-27 WO disclosed
US-20240352046-A1 ECTONUCLEOTIDE PYROPHOSPHATASE-PHOSPHODIESTERASE-1 (ENPP1) INHIBITORS AND USES THEREOF 1CBIO INC (US) 2024-10-24 US disclosed
US-20240139125-A1 BI-1 ANTAGONISTS AND THEIR USES INDUSTRIAL COOPERATION FOUNDATION JEONBUK NATIONAL UNIVERSITY (KR) 2024-05-02 US disclosed
CN-117800922-A SOS1 inhibitors 北京望实智慧科技有限公司 2024-04-02 CN disclosed
CN-117402143-A EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2024-01-16 CN disclosed
CN-117069700-A EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-11-17 CN disclosed
EP-0107398-B1 ORTHO SUBSTITUTED DIHYDROXY-2(1H)QUINAZOLINONE-1-ALKANOIC ACIDS ORTHO PHARMA CORP (US) 1988-06-08 EP disclosed
US-4645836-A Process for the preparation of 6,7-dihydroxy-4-alkyl-2(1H) quinazolinone-1-propionic acids ORTHO PHARMACEUTICAL CORPORATION (US) 1987-02-24 US disclosed
US-4631283-A RENAL VASODILATORS, CARDIOVASCULAR AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1986-12-23 US disclosed
US-4556739-A QUINAZOLINONE INTERMEDIATES ORTHO PHARMACEUTICAL CORPORATION (US) 1985-12-03 US disclosed
US-4555570-A Substituted 4-alkyl-2-(1H) quinazolinone-1-alkanoic acid derivatives ORTHO PHARMACEUTICAL CORPORATION (US) 1985-11-26 US disclosed
EP-0138492-A2 Process for preparing substituted 4-alkyl-2(1H) quinazolinone-1-alkanoic acid derivatives ORTHO PHARMACEUTICAL CORPORATION (US) 1985-04-24 EP disclosed
US-4490374-A CARDIOVASCULAR AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1984-12-25 US disclosed
EP-0107398-A1 Ortho substituted dihydroxy-2(1H)quinazolinone-1-alkanoic acids ORTHO PHARMACEUTICAL CORPORATION (US) 1984-05-02 EP disclosed
US-3987047-A ANORETICS BOEHRINGER INGELHEIM GMBH (DT) 1976-10-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260022135-A1 ECTONUCLEOTIDE PYROPHOSPHATASE-PHOSPHODIESTERASE-1 (ENPP1) INHIBITORS AND USES THEREOF ENPP1, ENPP3, NCEH1 KDM4E 4523/4885HTT 4450/4885CYP3A4 2626/4885
US-20240352046-A1 ECTONUCLEOTIDE PYROPHOSPHATASE-PHOSPHODIESTERASE-1 (ENPP1) INHIBITORS AND USES THEREOF ENPP1, ENPP3, ENPP2 KDM4E 3129/4885HTT 3735/4885CYP3A4 2491/4885
US-12325720-B2 Ectonucleotide pyrophosphatase-phosphodiesterase-1 (ENPP1) inhibitors and uses thereof ENPP1, ENPP3, ENPP2 KDM4E 3129/4885HTT 3735/4885CYP3A4 2491/4885
US-20240139125-A1 BI-1 ANTAGONISTS AND THEIR USES TMBIM6, RPS6KB1, RACK1 KDM4E 2423/4885HTT 3125/4885CYP3A4 4655/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.