SCHEMBL2176222

SCHEMBL2176222

CNC(=O)c1cc2cnccc2s1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 4/20 0.52
HDAC3 O15379 3/20 0.52
HDAC2 Q92769 3/20 0.52
NCOR2 Q9Y618 1/20 0.52
CYP2A6 P11509 4/20 0.51
CDK8 P49336 3/20 0.49
CHEK1 O14757 1/20 0.49
AURKA O14965 1/20 0.49
DAPK3 O43293 1/20 0.49
PRKD3 O94806 1/20 0.49
MAP4K4 O95819 1/20 0.49
PAK4 O96013 1/20 0.49
ABL1 P00519 1/20 0.49
RET P07949 1/20 0.49
PIM1 P11309 1/20 0.49
FGFR1 P11362 1/20 0.49
PRKACA P17612 1/20 0.49
FLT1 P17948 1/20 0.49
LTK P29376 1/20 0.49
GRK5 P34947 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7621269 0.88 CDK8 (0.65) CYP2A6CDK8CHEK1AURKADAPK3
SCHEMBL10857362 0.87 HDAC1 (0.60) HDAC1HDAC3HDAC2NCOR2CYP2A6
SCHEMBL10855370 0.84 HDAC1 (0.49) HDAC1HDAC3HDAC2NCOR2CYP2A6
SCHEMBL2009820 0.82 DYRK1A (0.56) HDAC1HDAC3HDAC2NCOR2CYP2A6
SCHEMBL160500 0.81 CDK8 (0.49) HDAC1HDAC3HDAC2NCOR2CYP2A6
SCHEMBL2012989 0.80 HDAC1 (0.54) HDAC1HDAC3HDAC2NCOR2CYP2A6
SCHEMBL844056 0.80 BCL2L1 (0.58) HDAC1HDAC3HDAC2NCOR2CYP2A6
SCHEMBL28769185 0.79 DAPK3 (0.76) HDAC1HDAC3HDAC2NCOR2CYP2A6
SCHEMBL2010041 0.78 HDAC1 (0.49) HDAC1HDAC3HDAC2NCOR2CYP2A6
SCHEMBL21470630 0.78 DYRK1A (0.49) HDAC1HDAC3HDAC2NCOR2CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079804-A1 CERTAIN TRIAZOLOPYRIDINES AND TRIAZOLOPYRAZINES, COMPOSITIONS THEREOF AND METHODS OF USE THEREFOR HUTCHISON MEDIPHARMA LIMITED (CN) 2011-07-07 WO disclosed