SCHEMBL21762403

SCHEMBL21762403

c1cnc2c(c1)SNCC1CCN21

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 17/20 0.47
HTR2C P28335 17/20 0.47
HTR2B P41595 17/20 0.47
CHRNA7 P36544 1/20 0.34
HTR3A P46098 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21762803 1.00 HTR2A (0.47) HTR2AHTR2CHTR2BCHRNA7HTR3A
SCHEMBL21762783 0.92 HTR2A (0.45) HTR2AHTR2CHTR2B
SCHEMBL21745067 0.90 HTR2A (0.44) HTR2AHTR2CHTR2B
SCHEMBL21745496 0.90 HTR2A (0.44) HTR2AHTR2CHTR2B
SCHEMBL21745068 0.90 HTR2A (0.44) HTR2AHTR2CHTR2B
SCHEMBL21745502 0.82 HTR2A (0.38) HTR2AHTR2CHTR2B
SCHEMBL21745501 0.82 HTR2A (0.38) HTR2AHTR2CHTR2B
SCHEMBL21745108 0.82 HTR2A (0.38) HTR2AHTR2CHTR2B
SCHEMBL21713741 0.69 HTR2A (0.45) HTR2AHTR2CHTR2BCHRNA7HTR3A
SCHEMBL21745092 0.69 HTR2A (0.45) HTR2AHTR2CHTR2BCHRNA7HTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3833662-B1 INHIBITORS OF KEAP1-NRF2 PROTEIN-PROTEIN INTERACTION JANSSEN PHARMACEUTICA NV (BE) 2024-01-17 EP disclosed
WO-2020041169-A2 INHIBITORS OF KEAP1-NRF2 PROTEIN-PROTEIN INTERACTION JANSSEN PHARMACEUTICA NV (BE) 2020-02-27 WO disclosed