SCHEMBL21764

SCHEMBL21764

Clc1ccccc1COc1cccc(OBOc2cccc(OCc3ccccc3Cl)c2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 3/20 0.58
NPC1 O15118 1/20 0.58
RAB9A P51151 1/20 0.58
MAOB P27338 3/20 0.50
MAOA P21397 1/20 0.50
SPHK2 Q9NRA0 2/20 0.46
SPHK1 Q9NYA1 2/20 0.46
IDO1 P14902 2/20 0.44
F9 P00740 1/20 0.44
NR1H2 P55055 1/20 0.44
NR1H3 Q13133 1/20 0.44
LMNA P02545 1/20 0.44
POLB P06746 1/20 0.44
GCK P35557 1/20 0.44
NR4A1 P22736 1/20 0.43
NR4A3 Q92570 1/20 0.43
TP53 P04637 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
AR P10275 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL791586 0.82 MAOB (0.60) NR4A2NPC1RAB9AMAOBMAOA
SCHEMBL257758 0.79 NR4A2 (0.60) NR4A2NPC1RAB9AMAOBMAOA
SCHEMBL4638867 0.79 MAOB (0.60) NR4A2NPC1RAB9AMAOBMAOA
SCHEMBL26377963 0.79 NR4A2 (0.60) NR4A2NPC1RAB9AMAOBMAOA
SCHEMBL12269215 0.79 NR4A2 (0.60) NR4A2NPC1RAB9AMAOBMAOA
SCHEMBL9812484 0.79 NR4A2 (0.69) NR4A2NPC1RAB9AMAOBMAOA
SCHEMBL23118 0.78 ABCB1 (0.53) MAOBSPHK2SPHK1IDO1F9
SCHEMBL7170719 0.77 NR4A2 (0.71) NR4A2NPC1RAB9AMAOBMAOA
SCHEMBL21762 0.76 NR4A2 (0.66) NR4A2NPC1RAB9AMAOBMAOA
SCHEMBL22316 0.76 MAOB (0.66) NR4A2MAOBMAOASPHK2SPHK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2609089-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2013-07-03 EP disclosed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed