SCHEMBL21769151

SCHEMBL21769151

CNc1ccc(Oc2ccnc3cc(OC)c(OC)cc23)cn1

nearest known ligand 0.74

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MET P08581 11/20 0.74
PDGFRB P09619 1/20 0.67
PDGFRA P16234 1/20 0.67
FGFR2 P21802 3/20 0.63
PTK2 Q05397 1/20 0.58
PTK2B Q14289 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22200852 0.87 MET (0.58) METPDGFRBPDGFRAFGFR2PTK2
SCHEMBL21769156 0.87 MET (0.71) METPDGFRBPDGFRAFGFR2
SCHEMBL22407346 0.87 MET (0.71) METPDGFRBPDGFRAFGFR2
SCHEMBL21966347 0.86 MET (1.00) METPDGFRA
SCHEMBL20782537 0.86 MET (0.69) METPDGFRBPDGFRAFGFR2
SCHEMBL21769367 0.85 PDGFRB (0.64) METPDGFRBPDGFRAFGFR2
SCHEMBL3904910 0.84 PDGFRA (0.70) METPDGFRBPDGFRAFGFR2
SCHEMBL7480761 0.84 FGFR2 (0.78) PDGFRBPDGFRAFGFR2
SCHEMBL3895466 0.84 PDGFRB (0.70) METPDGFRBPDGFRAFGFR2
SCHEMBL22703856 0.83 PDGFRB (0.68) METPDGFRBPDGFRAFGFR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3842425-A1 NOVEL QUINOLINE DERIVATIVE INHIBITOR Nanjing Transthera Biosciences Co., Ltd. (CN) 2021-06-30 EP disclosed
WO-2020141470-A1 QUINOLINE COMPOUNDS AS INHIBITORS OF TAM AND MET KINASES ARRAY BIOPHARMA INC. (US) 2020-07-09 WO disclosed
WO-2020038460-A1 NOVEL QUINOLINE DERIVATIVE INHIBITOR 南京药捷安康生物科技有限公司 2020-02-27 WO disclosed