SCHEMBL21770845

SCHEMBL21770845

CCCN(C)Cc1ccc(OC(CCNC)c2ccc(F)cc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 11/20 0.62
SLC6A2 P23975 3/20 0.47
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
LMNA P02545 4/20 0.46
CYP2D6 P10635 3/20 0.46
CYP2C19 P33261 3/20 0.46
NPC1 O15118 2/20 0.46
MTOR P42345 2/20 0.46
RAB9A P51151 2/20 0.46
CYP3A4 P08684 2/20 0.46
HTR2C P28335 2/20 0.46
SLC6A3 Q01959 2/20 0.46
CYP2C9 P11712 2/20 0.46
KDM4E B2RXH2 1/20 0.46
TP53 P04637 1/20 0.46
CYP1A2 P05177 1/20 0.46
ALOX15 P16050 1/20 0.46
TSHR P16473 1/20 0.46
NFKB1 P19838 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2615211 0.83 SLC6A4 (0.85) SLC6A4SLC6A2MEN1KMT2ALMNA
SCHEMBL2615212 0.83 SLC6A4 (0.85) SLC6A4SLC6A2MEN1KMT2ALMNA
SCHEMBL21770743 0.80 SLC6A4 (0.57) SLC6A4SLC6A2MEN1KMT2ALMNA
SCHEMBL21770733 0.79 SLC6A4 (0.57) SLC6A4SLC6A2MEN1KMT2ALMNA
SCHEMBL2615210 0.79 SLC6A4 (0.76) SLC6A4SLC6A2MEN1KMT2ALMNA
SCHEMBL2615209 0.77 SLC6A4 (1.00) SLC6A4SLC6A2MEN1KMT2ALMNA
SCHEMBL4740237 0.75 SLC6A4 (0.78) SLC6A4SLC6A2MEN1KMT2ALMNA
SCHEMBL15308539 0.75 PYCR1 (0.56) MEN1KMT2AKDM4ESIGMAR1HRH3
SCHEMBL9197291 0.74 SLC6A4 (0.61) SLC6A4SLC6A2MEN1KMT2ALMNA
SCHEMBL14566144 0.73 TAAR1 (0.55) MEN1KMT2ALMNARAB9ASIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3452475-B1 TETRAHYDROPYRIMIDODIAZEPINE AND TETRAHYDROPYRIDODIAZEPINE COMPOUNDS FOR TREATING PAIN AND PAIN RELATED CONDITIONS ESTEVE PHARMACEUTICALS SA (ES) 2020-02-26 EP disclosed