SCHEMBL21777144

SCHEMBL21777144

O=C(O)N(c1cscn1)S(=O)(=O)c1cnc(Cl)c(Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.46
NPSR1 Q6W5P4 4/20 0.46
MAPT P10636 1/20 0.35
TRPM8 Q7Z2W7 2/20 0.33
LMNA P02545 1/20 0.32
POLB P06746 1/20 0.32
JAK2 O60674 1/20 0.32
PKM P14618 1/20 0.32
SCN8A Q9UQD0 2/20 0.31
SCN1A P35498 1/20 0.31
SCN5A Q14524 1/20 0.31
L3MBTL1 Q9Y468 2/20 0.31
MAPK1 P28482 1/20 0.31
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21773513 0.88 ALDH1A1 (0.33) ALDH1A1NPSR1TRPM8SCN8ASCN1A
SCHEMBL30047031 0.84 ALDH1A1 (0.43) ALDH1A1NPSR1MAPTLMNAPOLB
SCHEMBL21783446 0.84 ALDH1A1 (0.43) ALDH1A1NPSR1MAPTLMNAPOLB
SCHEMBL21777235 0.81 ALDH1A1 (0.47) ALDH1A1MAPTTRPM8LMNAPOLB
SCHEMBL19613825 0.81 FLT1 (0.34) ALDH1A1MAPTTRPM8LMNASCN8A
SCHEMBL20449230 0.80 TDP1 (0.37) TRPM8SCN8ASCN1ASCN5ATDP1
SCHEMBL21777133 0.76 SCN1A (0.65) SCN8ASCN1ASCN5A
SCHEMBL21777131 0.76 SCN1A (0.65) SCN8ASCN1ASCN5A
SCHEMBL320178 0.74 SCN8A (0.36) SCN8ASCN1ASCN5A
SCHEMBL21783363 0.73 SCN8A (0.43) ALDH1A1NPSR1SCN8ASCN1ASCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11639351-B2 Heteroaryl-substituted sulfonamide compounds and their use as therapeutic agents XENON PHARMACEUTICALS INC. 2023-05-02 US disclosed
EP-3844150-A1 HETEROARYL-SUBSTITUTED SULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS Xenon Pharmaceuticals Inc. (CA) 2021-07-07 EP disclosed
US-10981905-B2 Heteroaryl-substituted sulfonamide compounds and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2021-04-20 US disclosed
US-20200157089-A1 HETEROARYL-SUBSTITUTED SULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2020-05-21 US disclosed
WO-2020047323-A1 HETEROARYL-SUBSTITUTED SULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2020-03-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11639351-B2 Heteroaryl-substituted sulfonamide compounds and their use as therapeutic agents SCN1A, SCN2A, SCN2B ALDH1A1 2781/4885NPSR1 455/4885MAPT 195/4885
US-20200157089-A1 HETEROARYL-SUBSTITUTED SULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS SCN1A, SCN2A, SCN2B ALDH1A1 2781/4885NPSR1 455/4885MAPT 195/4885
US-10981905-B2 Heteroaryl-substituted sulfonamide compounds and their use as therapeutic agents SCN1A, SCN2A, SCN2B ALDH1A1 2781/4885NPSR1 455/4885MAPT 195/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.