SCHEMBL21777869

SCHEMBL21777869

COc1ccc(Cn2nc(I)c3c(Oc4ccc(-c5cnn(-c6ccc(F)cc6)c(=O)c5C(N)=O)cc4F)ccnc32)cc1

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
F10 P00742 2/20 0.37
F2 P00734 1/20 0.37
CTRB1 P17538 1/20 0.37
NPBWR1 P48145 2/20 0.36
ALDH1A1 P00352 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
MET P08581 14/20 0.36
AXL P30530 10/20 0.36
MERTK Q12866 9/20 0.36
TYRO3 Q06418 8/20 0.36
MST1R Q04912 1/20 0.35
MAPKAPK2 P49137 1/20 0.34
MCHR1 Q99705 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4722856 0.86 PDE1B (0.37) F10F2CTRB1ALDH1A1MET
SCHEMBL30693661 0.80 AXL (0.58) METAXLMERTKTYRO3
SCHEMBL3103995 0.80 AXL (0.58) METAXLMERTKTYRO3
SCHEMBL30208939 0.77 AXL (0.57) METAXLMERTKTYRO3
SCHEMBL21785971 0.77 AXL (0.57) METAXLMERTKTYRO3
SCHEMBL1944519 0.75 AXL (0.38) METAXL
SCHEMBL3106815 0.74 MET (0.59) METMST1R
SCHEMBL3104308 0.74 AXL (0.57) METAXLMERTKTYRO3
SCHEMBL3103490 0.74 AXL (0.44) METAXLMERTKTYRO3
SCHEMBL3101305 0.73 MET (0.39) METAXLMERTKTYRO3MST1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3843850-A1 PYRAZOLO[3,4-B]PYRIDINE COMPOUNDS AS INHIBITORS OF TAM AND MET KINASES Array BioPharma Inc. (US) 2021-07-07 EP disclosed
WO-2020047184-A1 PYRAZOLO[3,4-b]PYRIDINE COMPOUNDS AS INHIBITORS OF TAM AND MET KINASES ARRAY BIOPHARMA INC. (US) 2020-03-05 WO disclosed