SCHEMBL21779374

SCHEMBL21779374

Cc1ccc(CNc2ncc(-c3cnn(C)c3)cc2C(N)=O)cc1C

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RPS6KB1 P23443 2/20 0.55
PDPK1 O15530 1/20 0.55
AXL P30530 5/20 0.53
MERTK Q12866 5/20 0.53
MET P08581 6/20 0.50
JAK2 O60674 2/20 0.45
JAK1 P23458 2/20 0.45
JAK3 P52333 2/20 0.45
TYK2 P29597 1/20 0.45
IKBKE Q14164 1/20 0.43
TBK1 Q9UHD2 1/20 0.43
GHSR Q92847 2/20 0.42
MKNK1 Q9BUB5 1/20 0.42
MKNK2 Q9HBH9 1/20 0.42
KCNH2 Q12809 1/20 0.42
ATM Q13315 1/20 0.42
ATR Q13535 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18580740 0.91 AXL (0.51) RPS6KB1PDPK1AXLMERTKMET
SCHEMBL18616235 0.81 PDPK1 (0.48) RPS6KB1PDPK1METJAK2JAK3
SCHEMBL18580289 0.76 MERTK (0.72) AXLMERTKMET
SCHEMBL663299 0.71 RPS6KB1 (1.00) RPS6KB1PDPK1
SCHEMBL18611803 0.71 IKBKE (0.62) AXLMERTKMETIKBKETBK1
SCHEMBL30108229 0.71 IKBKE (0.62) AXLMERTKMETIKBKETBK1
SCHEMBL18580676 0.71 MET (0.46) AXLMERTKMETIKBKETBK1
SCHEMBL18615746 0.71 RPS6KB1 (0.48) RPS6KB1
SCHEMBL18580544 0.69 AXL (1.00) AXLMERTKMET
SCHEMBL18580541 0.69 AXL (1.00) AXLMERTKMET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3344613-B1 HETEROARYL COMPOUNDS AND THEIR USE AS THERAPEUTIC DRUGS DONG A SOCIO HOLDINGS CO LTD (KR) 2020-03-04 EP disclosed