SCHEMBL21780682

SCHEMBL21780682

CCc1ccc(SN(C)C)cc1C(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AR P10275 5/20 0.37
POLQ O75417 9/20 0.36
IDO1 P14902 2/20 0.36
SLC6A4 P31645 3/20 0.32
SLC6A2 P23975 2/20 0.32
EPHX2 P34913 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19145665 0.77 AR (0.38) AR
SCHEMBL21516362 0.74 CRHR1 (0.48) ARPOLQ
SCHEMBL20388971 0.73 NOTUM (0.39) AR
SCHEMBL12834802 0.71 FFAR4 (0.40) ARIDO1EPHX2
SCHEMBL4416164 0.71 POLQ (0.51) POLQIDO1
SCHEMBL10256179 0.71 SMN1; SMN2 (0.39) ARPOLQIDO1EPHX2
SCHEMBL8417818 0.71 IDO1 (0.59) POLQIDO1SLC6A4SLC6A2EPHX2
SCHEMBL16770736 0.69 KDM1A (0.42) ARPOLQIDO1SLC6A4EPHX2
SCHEMBL19304121 0.69 HSD17B3 (0.41) ARPOLQIDO1EPHX2
SCHEMBL805479 0.69 POLQ (0.52) POLQSLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3722284-A1 3-((HETERO-)ARYL)-8-AMINO-2-OXO-1,3-DIAZA-SPIRO-[4.5]-DECANE DERIVATIVES Grünenthal GmbH (DE) 2020-10-14 EP disclosed
EP-3402781-B1 3-((HETERO-)ARYL)-8-AMINO-2-OXO-1,3-DIAZA-SPIRO-[4.5]-DECANE DERIVATIVES GRUENENTHAL GMBH (DE) 2020-03-04 EP disclosed