SCHEMBL21780776

SCHEMBL21780776

COCOc1ccc(C(=O)Cc2ccc(OC)cc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.60
HTT P42858 3/20 0.60
LMNA P02545 1/20 0.60
MAPT P10636 2/20 0.55
KMT2A Q03164 1/20 0.55
RAB9A P51151 2/20 0.53
POLB P06746 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
GSK3B P49841 1/20 0.51
HDAC3 O15379 1/20 0.51
HDAC4 P56524 1/20 0.51
HDAC1 Q13547 1/20 0.51
HDAC7 Q8WUI4 1/20 0.51
HDAC2 Q92769 1/20 0.51
HDAC10 Q969S8 1/20 0.51
HDAC11 Q96DB2 1/20 0.51
HDAC8 Q9BY41 1/20 0.51
HDAC6 Q9UBN7 1/20 0.51
HDAC9 Q9UKV0 1/20 0.51
HDAC5 Q9UQL6 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17845146 0.89 NPC1 (0.55) NPC1HTTLMNAMAPTKMT2A
SCHEMBL457954 0.88 NPC1 (0.73) NPC1HTTLMNAMAPTKMT2A
SCHEMBL1515877 0.88 STS (0.56) NPC1HTTLMNAMAPTRAB9A
SCHEMBL21780777 0.85 POLB (0.55) NPC1HTTLMNAMAPTKMT2A
SCHEMBL12188828 0.83 MAPT (0.62) NPC1HTTLMNAMAPTKMT2A
SCHEMBL2938988 0.82 NPC1 (0.42) NPC1HTTLMNAMAPTKMT2A
SCHEMBL3099733 0.82 NPC1 (0.65) NPC1HTTLMNAMAPTKMT2A
SCHEMBL1420182 0.82 NPC1 (0.65) NPC1HTTLMNAMAPTKMT2A
SCHEMBL3097303 0.82 NPC1 (0.65) NPC1HTTLMNAMAPTKMT2A
SCHEMBL12637609 0.82 NPC1 (0.65) NPC1HTTLMNAMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233828-B1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF HOFFMANN LA ROCHE (CH) 2020-03-04 EP disclosed