SCHEMBL21780867

SCHEMBL21780867

C=Cc1ccc(-c2ccccc2)c(C=CC)c1C

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 1/20 0.32
AKT2 P31751 1/20 0.32
ESR2 Q92731 1/20 0.32
PSMB5 P28074 1/20 0.31
PDCD1 Q15116 1/20 0.31
CD274 Q9NZQ7 1/20 0.31
CYP2A6 P11509 1/20 0.30
CYP2B6 P20813 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16296809 0.81 ESR2 (0.40) AKT1AKT2ESR2PDCD1CD274
SCHEMBL29114020 0.74 PARP10 (0.39) AKT1AKT2ESR2PSMB5PDCD1
SCHEMBL8848267 0.73 ALDH1A1 (0.37) CYP2A6
SCHEMBL22255953 0.73
SCHEMBL31432621 0.73 ALDH1A1 (0.37) CYP2A6
SCHEMBL21636879 0.72
SCHEMBL7550211 0.72 PDCD1 (0.48) AKT1AKT2PSMB5PDCD1CD274
SCHEMBL25330371 0.70 BRD4 (0.36) AKT2
SCHEMBL6548166 0.70 KDM4E (0.40) ESR2PDCD1CD274CYP2A6CYP2B6
SCHEMBL27898117 0.70 ALDH1A1 (0.43) ESR2CYP2A6CYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233828-B1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF HOFFMANN LA ROCHE (CH) 2020-03-04 EP disclosed