SCHEMBL217811

SCHEMBL217811

CN(C[C@H]1CC(=O)[C@@]2(C)CCC3c4ccc(O)cc4CCC3C12)S(=O)(=O)c1ccc2ccccc2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STS P08842 10/20 0.53
ESR1 P03372 6/20 0.47
ESR2 Q92731 4/20 0.47
HSD17B1 P14061 2/20 0.47
AKR1B10 O60218 1/20 0.47
LMNA P02545 1/20 0.47
SHBG P04278 1/20 0.47
CYP1A2 P05177 1/20 0.47
PGR P06401 1/20 0.47
SERPINA6 P08185 1/20 0.47
CYP3A4 P08684 1/20 0.47
AR P10275 1/20 0.47
MAPT P10636 1/20 0.47
CYP19A1 P11511 1/20 0.47
AKR1B1 P15121 1/20 0.47
NFKB1 P19838 1/20 0.47
SLC6A4 P31645 1/20 0.47
OPRM1 P35372 1/20 0.47
SNCA P37840 1/20 0.47
HTR2B P41595 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2738663 1.00 STS (0.53) STSESR1ESR2HSD17B1AKR1B10
SCHEMBL217882 0.92 STS (0.50) STSESR1ESR2HSD17B1AKR1B10
SCHEMBL217881 0.92 STS (0.50) STSESR1ESR2HSD17B1AKR1B10
SCHEMBL218444 0.89 STS (0.51) STSESR1ESR2HSD17B1AKR1B10
SCHEMBL218899 0.89 STS (0.51) STSESR1ESR2HSD17B1AKR1B10
SCHEMBL218445 0.89 STS (0.51) STSESR1ESR2HSD17B1AKR1B10
SCHEMBL218900 0.89 STS (0.51) STSESR1ESR2HSD17B1AKR1B10
SCHEMBL219426 0.89 HSD17B1 (0.49) STSESR1ESR2HSD17B1AKR1B10
SCHEMBL219425 0.89 HSD17B1 (0.49) STSESR1ESR2HSD17B1AKR1B10
SCHEMBL218082 0.88 STS (0.51) STSESR1ESR2HSD17B1AKR1B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088758-B2 17β-hydroxysteroid dehydrogenase type I inhibitors ABBOTT PRODUCTS GMBH (DE) 2012-01-03 US claimed
US-8088758-B2 17β-hydroxysteroid dehydrogenase type I inhibitors ABBOTT PRODUCTS GMBH (DE) 2012-01-03 US disclosed