SCHEMBL21782467

SCHEMBL21782467

Cc1cc(F)ccc1C(C)(C)O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.42
HDAC3 O15379 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC2 Q92769 1/20 0.42
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
NR3C1 P04150 4/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
CHRM3 P20309 1/20 0.35
PTGS1 P23219 3/20 0.34
PTGS2 P35354 3/20 0.34
NR3C2 P08235 2/20 0.34
MCL1 Q07820 1/20 0.34
ACHE P22303 2/20 0.33
CA3 P07451 1/20 0.33
CA6 P23280 1/20 0.33
CA5A P35218 1/20 0.33
CA9 Q16790 1/20 0.33
CA14 Q9ULX7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18711606 0.83 NR3C1 (0.44) MEN1KMT2ANR3C1CHRM3NR3C2
SCHEMBL9607555 0.82 HDAC6 (0.41) HDAC6HDAC3HDAC1HDAC2TSHR
SCHEMBL18802727 0.82 MEN1 (0.42) MEN1KMT2ANR3C1CHRM3PTGS1
SCHEMBL1507033 0.80 KCNN4 (0.43) HDAC6HDAC3HDAC1HDAC2MEN1
SCHEMBL29727285 0.80 KCNN4 (0.43) HDAC6HDAC3HDAC1HDAC2MEN1
SCHEMBL10035077 0.80 HDAC6 (0.40) HDAC6HDAC3HDAC1HDAC2NR3C1
SCHEMBL21916381 0.78 HDAC6 (0.39) HDAC6HDAC3HDAC1HDAC2NR3C1
SCHEMBL18701599 0.78 PTGS1 (0.42) MEN1KMT2ANR3C1TSHRPTGS1
SCHEMBL12180439 0.77 TDP1 (0.46) MEN1KMT2AALDH1A1MAPT
SCHEMBL9272585 0.77 ESR1 (0.41) MEN1KMT2ATSHRALDH1A1TNKS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3407877-B1 NLRP3 INHIBITORS FOR THE TREATMENT OF INFLAMMATORY SKIN DISORDERS GALDERMA RES & DEV (FR) 2020-03-04 EP disclosed