SCHEMBL21782876

SCHEMBL21782876

C=C/C=C\C=C(/N)NC(=O)CCC

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSD P07339 1/20 0.39
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
MAPT P10636 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
THRB P10828 1/20 0.33
FAAH O00519 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CASP2 P42575 1/20 0.31
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22540311 0.80 CTSD (0.37) CTSDHDAC3HDAC1HDAC2HDAC8
SCHEMBL13522735 0.70 KDM4A (0.30)
SCHEMBL20157549 0.69 HDAC3 (0.40) CTSDHDAC3HDAC1HDAC2HDAC8
SCHEMBL4879049 0.68
SCHEMBL2933109 0.67 HDAC3 (0.46) CTSDHDAC3HDAC1HDAC2HDAC8
SCHEMBL1643947 0.67 HDAC3 (0.63) CTSDHDAC3HDAC1HDAC2HDAC8
SCHEMBL22540338 0.66 HDAC3 (0.36) CTSDHDAC3HDAC1HDAC2HDAC8
Water SCHEMBL29155573 0.65 HDAC3 (0.60) CTSDHDAC3HDAC1HDAC2HDAC8
SCHEMBL14291827 0.65 FFAR3 (0.31) HDAC3HDAC1HDAC2HDAC8
SCHEMBL8293489 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3402783-B1 3-(CARBOXYETHYL)-8-AMINO-2-OXO-1,3-DIAZA-SPIRO-[4.5]-DECANE DERIVATIVES GRUENENTHAL GMBH (DE) 2020-03-04 EP disclosed