SCHEMBL21783201

SCHEMBL21783201

COc1c(N2CCN(C(=O)OC(C)(P(=O)(O)O)P(=O)(O)O)C(C)C2)c(C)c(N)c2c(=O)c(C(=O)O)cn(C3CC3)c12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.49
HPGD P15428 3/20 0.49
ALDH1A1 P00352 3/20 0.49
LMNA P02545 2/20 0.49
CYP2C19 P33261 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
ATM Q13315 1/20 0.45
POLB P06746 3/20 0.45
TDP1 Q9NUW8 3/20 0.45
NPSR1 Q6W5P4 1/20 0.45
KCNH2 Q12809 6/20 0.43
CACNA1F O60840 1/20 0.43
MAPK1 P28482 1/20 0.43
CACNA1D Q01668 1/20 0.43
CACNA1S Q13698 1/20 0.43
CACNA1C Q13936 1/20 0.43
PRKD3 O94806 1/20 0.42
ALOX15 P16050 1/20 0.42
OPRM1 P35372 1/20 0.42
CLK2 P49760 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22778992 0.92 KDM4E (0.52) KDM4EHPGDALDH1A1LMNACYP2C19
SCHEMBL21783269 0.88 KDM4E (0.51) KDM4EHPGDALDH1A1LMNACYP2C19
SCHEMBL23197070 0.80 KDM4E (0.54) KDM4EHPGDALDH1A1LMNACYP2C19
SCHEMBL26931416 0.77 CACNA1F (0.65) POLBKCNH2CACNA1FMAPK1CACNA1D
SCHEMBL22778993 0.77 KCNH2 (0.62) KDM4EHPGDALDH1A1LMNACYP2C19
SCHEMBL21074735 0.76 KDM4E (0.49) KDM4EHPGDALDH1A1LMNACYP2C19
SCHEMBL5003903 0.75 KDM4E (0.75) KDM4EHPGDALDH1A1LMNACYP2C19
SCHEMBL26932000 0.74 KDM4E (0.47) KDM4EHPGDALDH1A1LMNACYP2C19
SCHEMBL21074775 0.72 MEN1 (0.65) KDM4EHPGDALDH1A1LMNAPOLB
SCHEMBL8564558 0.72 KCNH2 (0.57) KDM4EHPGDALDH1A1LMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020014269-A9 BISPHOSPHONATE QUINOLONE CONJUGATES AND USES THEREOF BIOVINC, LLC. (US) 2020-03-05 WO disclosed