SCHEMBL21784837

SCHEMBL21784837

Clc1ccc(CCn2ccnn2)c(Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.46
CCR1 P32246 8/20 0.45
CCR2 P41597 8/20 0.45
CCR4 P51679 6/20 0.45
CYP3A4 P08684 3/20 0.44
CYP2C9 P11712 3/20 0.44
CYP2C19 P33261 2/20 0.44
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
DAO P14920 1/20 0.43
IDO1 P14902 1/20 0.41
PSEN1 P49768 1/20 0.40
PSEN2 P49810 1/20 0.40
APH1B Q8WW43 1/20 0.40
NCSTN Q92542 1/20 0.40
APH1A Q96BI3 1/20 0.40
PSENEN Q9NZ42 1/20 0.40
CYP19A1 P11511 3/20 0.40
CYP1A2 P05177 1/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7023638 0.78 KMT2A (0.46) KMT2ACYP3A4CYP2C9CYP2C19MAOA
SCHEMBL28761316 0.76 PSEN1 (0.37) KMT2ACCR1CCR2CCR4CYP3A4
SCHEMBL14370854 0.72 KDM4E (0.50) KMT2ACCR1CCR2CCR4CYP3A4
SCHEMBL5301838 0.72 CCR1 (0.54) CCR1CCR2CCR4CYP3A4CYP2C9
SCHEMBL8908893 0.72 CYP2C9 (0.54) KMT2ACYP3A4CYP2C9CYP2C19MAOA
SCHEMBL25934781 0.71 CYP19A1 (0.46) CCR1CCR2CCR4PSEN1PSEN2
SCHEMBL11621292 0.71 IDO1 (0.65) CYP3A4CYP2C9CYP2C19MAOAMAOB
SCHEMBL10851275 0.70 ALDH1A1 (0.53) KMT2ACYP19A1MAPK1LMNAHTT
SCHEMBL9657759 0.70 CYP3A4 (0.40) CCR1CCR2CCR4CYP3A4CYP2C9
SCHEMBL21784834 0.68 CYP3A4 (0.46) CCR1CCR2CCR4CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200072711-A1 FLUORESCENT ENDOPLASMIC RETICULUM TRACKERS FOR LIVE CELL IMAGING OF PATHOGENIC YEAST RAMOT AT TEL AVIV UNIVERSITY LTD. (IL) 2020-03-05 US disclosed