SCHEMBL21784994

SCHEMBL21784994

Fc1ccc(C2CCC(F)(F)CC2)c(Br)c1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNA4 P43681 1/20 0.35
OPRL1 P41146 11/20 0.35
HTR1A P08908 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
KDM1A O60341 2/20 0.32
GRM5 P41594 1/20 0.31
HTR2C P28335 1/20 0.31
HTR6 P50406 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19682735 0.85 CHRNB2 (0.41) CHRNB2CHRNB4CHRNA3CHRNA4OPRL1
SCHEMBL31071936 0.85 CHRNB2 (0.41) CHRNB2CHRNB4CHRNA3CHRNA4OPRL1
SCHEMBL21767543 0.76 BACE1 (0.33)
SCHEMBL31071957 0.76 BACE1 (0.33)
SCHEMBL21784957 0.76 ESR2 (0.37) CHRNB2CHRNB4CHRNA3CHRNA4OPRL1
SCHEMBL27797108 0.71 CHRNB2 (0.49) CHRNB2CHRNB4CHRNA3CHRNA4HTR1A
SCHEMBL24215291 0.69 QPCT (0.36) CHRNB2CHRNA4OPRL1KDM1A
SCHEMBL1782611 0.69 TP53 (0.42) CHRNB2CHRNB4CHRNA3CHRNA4HTR2C
SCHEMBL26615751 0.69 HDAC1 (0.32)
SCHEMBL21767694 0.68 OPRL1 (0.33) OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020047239-A1 INHIBITING αV β6 INTEGRIN MORPHIC THERAPEUTIC, INC. (US) 2020-03-05 WO disclosed