SCHEMBL21787685

SCHEMBL21787685

CCOC(=O)C1CN(Cc2ccccc2)C(C)CN1Cc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.51
PDK2 Q15119 1/20 0.51
PDK3 Q15120 1/20 0.51
PDK4 Q16654 1/20 0.51
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
MAPT P10636 1/20 0.49
TSHR P16473 1/20 0.47
POLB P06746 1/20 0.47
ALDH1A1 P00352 5/20 0.46
ATM Q13315 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
KDM4E B2RXH2 1/20 0.46
MAPK1 P28482 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
TRPC5 Q9UL62 1/20 0.44
MAPK14 Q16539 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11147455 0.93 MEN1 (0.55) MEN1KMT2APOLBALDH1A1ATM
SCHEMBL124103 0.82 L3MBTL1 (0.55) MEN1KMT2APOLBALDH1A1ATM
SCHEMBL3309475 0.82 MEN1 (0.54) MEN1KMT2ATSHRPOLBALDH1A1
SCHEMBL3306018 0.82 MEN1 (0.54) MEN1KMT2ATSHRPOLBALDH1A1
SCHEMBL8269795 0.81 MEN1 (0.50) MEN1KMT2AMAPTPOLBALDH1A1
SCHEMBL4662072 0.81 MEN1 (0.50) MEN1KMT2AMAPTPOLBALDH1A1
SCHEMBL5568190 0.81 MEN1 (0.50) MEN1KMT2AMAPTPOLBALDH1A1
SCHEMBL31309182 0.81 MEN1 (0.50) MEN1KMT2AMAPTPOLBALDH1A1
SCHEMBL5568192 0.81 MEN1 (0.50) MEN1KMT2AMAPTPOLBALDH1A1
SCHEMBL5373647 0.81 MAPT (0.51) MEN1KMT2AMAPTTSHRPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11001570-B2 6-amino-quinolinone compounds and derivatives as BCL6 inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2021-05-11 US disclosed
EP-3555063-B1 6-AMINO-QUINOLINONE COMPOUNDS AND DERIVATIVES AS BCL6 INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2020-09-16 EP disclosed
US-20200071297-A1 NEW 6-AMINO-QUINOLINONE COMPOUNDS AND DERIVATIVES AS BCL6 INHIBITORS BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2020-03-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200071297-A1 NEW 6-AMINO-QUINOLINONE COMPOUNDS AND DERIVATIVES AS BCL6 INHIBITORS BCL6, BCL6B, BCOR PDK1 1506/4885PDK2 2323/4885PDK3 1975/4885
US-11001570-B2 6-amino-quinolinone compounds and derivatives as BCL6 inhibitors BCL6, BCL6B, BCOR PDK1 1498/4885PDK2 2141/4885PDK3 1894/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.