SCHEMBL21790488

SCHEMBL21790488

CCCC(C)(C)Nc1cccc(C(=O)O)c1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.48
RAB9A P51151 3/20 0.48
ALDH1A1 P00352 2/20 0.48
POLB P06746 1/20 0.48
AKR1C3 P42330 2/20 0.48
NR1H4 Q96RI1 6/20 0.47
SMN1; SMN2 Q16637 2/20 0.46
MITF O75030 1/20 0.46
PAX8 Q06710 1/20 0.46
HIF1A Q16665 1/20 0.45
EPAS1 Q99814 1/20 0.45
AKR1C2 P52895 1/20 0.44
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13996668 0.88 NPC1 (0.50) NPC1RAB9AALDH1A1POLBAKR1C3
SCHEMBL23343714 0.85 NPC1 (0.46) NPC1RAB9AALDH1A1POLBAKR1C3
SCHEMBL2724979 0.84 NPC1 (0.55) NPC1RAB9AALDH1A1POLBAKR1C3
SCHEMBL14269924 0.77 RAB9A (0.49) NPC1RAB9AALDH1A1POLBAKR1C3
SCHEMBL1453847 0.76 GAA (0.43) ALDH1A1KMT2A
SCHEMBL23084782 0.76 MAPT (0.48) ALDH1A1POLBKMT2AMEN1
SCHEMBL21790803 0.74 EPHX1 (0.42) ALDH1A1POLBSMN1; SMN2KMT2AMEN1
SCHEMBL21799923 0.74 MAPT (0.43) ALDH1A1SMN1; SMN2KMT2AMEN1
SCHEMBL22600368 0.74 GAA (0.46) RAB9AALDH1A1SMN1; SMN2KMT2AMEN1
SCHEMBL873032 0.74 AKR1C3 (0.61) NPC1RAB9AALDH1A1AKR1C3NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200071308-A1 Benzene, Pyridine, and Pyridazine Derivatives ESANEX INC (US) 2020-03-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200071308-A1 Benzene, Pyridine, and Pyridazine Derivatives CDK4, P2RX4, MKI67 NPC1 4242/4885RAB9A 3778/4885ALDH1A1 1049/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.