SCHEMBL2182018

SCHEMBL2182018

CN(C)C(=O)c1ccc(Oc2ccc3c(c2)S(O)(O)NCN3C2CC2)cc1

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GRIA2 P42262 15/20 0.59
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
GRIA1 P42261 2/20 0.39
GRIA3 P42263 2/20 0.39
GRIA4 P48058 2/20 0.39
MMP13 P45452 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2182022 0.90 GRIA2 (0.71) GRIA2ALDH1A1HPGDSMN1; SMN2GRIA1
SCHEMBL2178746 0.78 GRIA2 (0.58) GRIA2GRIA1GRIA3GRIA4MMP13
SCHEMBL2161137 0.78 GRIA2 (0.62) GRIA2GRIA1GRIA3GRIA4
SCHEMBL2183670 0.77 GRIA2 (0.58) GRIA2ALDH1A1HPGDSMN1; SMN2GRIA1
SCHEMBL2152080 0.74 GRIA2 (1.00) GRIA2GRIA1GRIA3GRIA4
SCHEMBL2183726 0.74 GRIA2 (0.77) GRIA2GRIA1GRIA3GRIA4
SCHEMBL5620058 0.73 GRIA2 (0.41) GRIA2ALDH1A1HPGDSMN1; SMN2
SCHEMBL2152051 0.72 GRIA2 (1.00) GRIA2GRIA1GRIA3GRIA4
SCHEMBL5621550 0.71 GRIA2 (0.39) GRIA2ALDH1A1HPGD
SCHEMBL2179977 0.71 GRIA2 (1.00) GRIA2GRIA1GRIA3GRIA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011083265-A1 NOVEL DERIVATIVES OF CYCLOPROPYLATED BENZOTHIADIAZINES, METHOD FOR PREPARING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME LES LABORATOIRES SERVIER (FR) 2011-07-14 WO disclosed