SCHEMBL21822124

SCHEMBL21822124

N#Cc1ccc2cc(C(=O)O)n(CCc3ccccc3)c2c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR9 P51686 2/20 0.58
CCR2 P41597 5/20 0.52
PLA2G10 O15496 1/20 0.49
PLA2G2A P14555 1/20 0.49
ALDH1A1 P00352 2/20 0.47
CYP1A2 P05177 1/20 0.47
POLB P06746 1/20 0.47
HDAC8 Q9BY41 2/20 0.47
HDAC6 Q9UBN7 2/20 0.47
HDAC1 Q13547 1/20 0.47
NTRK1 P04629 1/20 0.47
GPR35 Q9HC97 1/20 0.46
KDM4E B2RXH2 2/20 0.46
TSHR P16473 2/20 0.46
HSD17B10 Q99714 2/20 0.46
GLA P06280 1/20 0.46
HPGD P15428 1/20 0.46
HTT P42858 1/20 0.46
MCL1 Q07820 2/20 0.43
ALB P02768 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31689701 1.00 CCR9 (0.58) CCR9CCR2PLA2G10PLA2G2AALDH1A1
SCHEMBL21822198 0.85 TSHR (0.53) CCR9PLA2G10PLA2G2AALDH1A1POLB
SCHEMBL1422436 0.82 CCR2 (0.74) CCR2PLA2G10ALDH1A1CYP1A2POLB
SCHEMBL31689681 0.81 CCR9 (0.52) CCR9CCR2PLA2G10PLA2G2AALDH1A1
SCHEMBL21822478 0.81 CCR9 (0.52) CCR9CCR2PLA2G10PLA2G2AALDH1A1
SCHEMBL21822281 0.81 CCR9 (0.69) CCR9CCR2GPR35
SCHEMBL31689688 0.81 CCR9 (0.69) CCR9CCR2GPR35
SCHEMBL28593764 0.81 CCR9 (0.72) CCR9CCR2GPR35
SCHEMBL21822343 0.80 F10 (0.49) CCR9PLA2G10PLA2G2AALDH1A1POLB
SCHEMBL10022666 0.80 CCR9 (0.65) CCR9CCR2PLA2G10PLA2G2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3860636-A1 MATRIPTASE 2 INHIBITORS AND USES THEREOF Disc Medicine, Inc. (US) 2021-08-11 EP disclosed
WO-2020072580-A1 MATRIPTASE 2 INHIBITORS AND USES THEREOF DISC MEDICINE, INC. (US) 2020-04-09 WO disclosed