SCHEMBL2183259

SCHEMBL2183259

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nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BMP1 P13497 3/20 0.45
DPP4 P27487 2/20 0.42
DPP8 Q6V1X1 2/20 0.42
DPP9 Q86TI2 2/20 0.42
BACE1 P56817 12/20 0.40
CTSD P07339 4/20 0.40
ALOX15 P16050 1/20 0.38
BLM P54132 1/20 0.38
PMP22 Q01453 1/20 0.38
KMT2A Q03164 1/20 0.38
GRM8 O00222 1/20 0.36
GRM6 O15303 1/20 0.36
GRIN2D O15399 1/20 0.36
GRIN3B O60391 1/20 0.36
GSR P00390 1/20 0.36
CYP1A2 P05177 1/20 0.36
GRIK1 P39086 1/20 0.36
GRM5 P41594 1/20 0.36
GRIA1 P42261 1/20 0.36
GRIA2 P42262 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2195933 0.95 BMP1 (0.42) BMP1DPP4DPP8DPP9BACE1
SCHEMBL2198349 0.95 DPP4 (0.46) BMP1DPP4DPP8DPP9BACE1
SCHEMBL2190812 0.95 DPP4 (0.46) BMP1DPP4DPP8DPP9BACE1
SCHEMBL2194678 0.92 BMP1 (0.44) BMP1DPP4DPP8DPP9BACE1
SCHEMBL2182643 0.90 BMP1 (0.45) BMP1DPP4DPP8DPP9BACE1
SCHEMBL2195713 0.90 DPP4 (0.43) BMP1DPP4DPP8DPP9BACE1
SCHEMBL7886832 0.89 DPP4 (0.46) BMP1DPP4DPP8DPP9BACE1
SCHEMBL11136056 0.88 DPP4 (0.51) BMP1DPP4DPP8DPP9BACE1
SCHEMBL2182616 0.87 DPP4 (0.46) BMP1DPP4DPP8DPP9BACE1
SCHEMBL2182958 0.86 DPP4 (0.48) BMP1DPP4DPP8DPP9BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110166063-A1 POLYMER CONJUGATES OF THERAPEUTIC PEPTIDES NEKTAR THERAPEUTICS (US) 2011-07-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110166063-A1 POLYMER CONJUGATES OF THERAPEUTIC PEPTIDES NGLY1, CD44, IAPP BMP1 3740/4885DPP4 525/4885DPP8 644/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.