SCHEMBL2183291

SCHEMBL2183291

Cc1c[c]cc(-c2ccc3[nH]ccc3c2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.53
BRD4 O60885 1/20 0.46
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA9 Q16790 1/20 0.45
PTGS2 P35354 1/20 0.44
CYP17A1 P05093 1/20 0.43
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
FYN P06241 1/20 0.41
IMPDH2 P12268 1/20 0.41
IMPDH1 P20839 1/20 0.41
NISCH Q9Y2I1 1/20 0.41
AHR P35869 3/20 0.41
NR4A2 P43354 2/20 0.41
CYP2A6 P11509 1/20 0.41
F7 P08709 1/20 0.41
LTA4H P09960 1/20 0.41
F3 P13726 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27461448 0.81 NPC1 (0.61) NPC1BRD4CA12CA1CA2
SCHEMBL31504064 0.81 NPC1 (0.61) NPC1BRD4CA12CA1CA2
SCHEMBL731092 0.80 NPC1 (0.49) NPC1BRD4CA12CA1CA2
SCHEMBL15296270 0.79 NPC1 (0.69) NPC1BRD4CA12CA1CA2
SCHEMBL5850255 0.78 NPC1 (0.79) NPC1BRD4CA12CA1CA2
SCHEMBL9231655 0.78 NPC1 (0.68) NPC1BRD4CA12CA1CA2
SCHEMBL732779 0.75 NPC1 (0.64) NPC1CA12CA1CA2CA9
SCHEMBL13354456 0.74 PIP4K2A (0.58) NPC1BRD4CA12CA1CA2
SCHEMBL732897 0.74 NPC1 (0.67) NPC1BRD4CA12CA1CA2
SCHEMBL2192638 0.73 NPC1 (0.47) NPC1BRD4CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110166132-A1 Gamma Secretase Modulators AMGEN INC. (US) 2011-07-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110166132-A1 Gamma Secretase Modulators BACE1, BACE2, PSEN1 NPC1 746/4885BRD4 1253/4885CA12 3978/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.