SCHEMBL218355

SCHEMBL218355

C1=Cc2ncncc2OC1

nearest known ligand 0.32

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.32
CA9 Q16790 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28972632 0.71 CA1 (0.31) CA1CA9
SCHEMBL3014139 0.69 HTT (0.31) CA1CA9
SCHEMBL160028 0.68 CA1 (0.34) CA1CA9
SCHEMBL1501891 0.68 CA1 (0.32) CA1CA9
SCHEMBL3605917 0.68 CA1 (0.32) CA1CA9
SCHEMBL28412569 0.67 CYP1A2 (0.37)
SCHEMBL30023511 0.67 CYP1A2 (0.34)
SCHEMBL3012197 0.66
SCHEMBL29955980 0.66
SCHEMBL218307 0.64

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 94 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119161353-A Design, synthesis and activity evaluation of pyranopyrimidine heterocyclic p97/VCP inhibitors 首都医科大学 2024-12-20 CN claimed
EP-1663993-B1 GUANIDINE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2008-03-12 EP claimed
US-20070123510-A1 Guanidine derivatives ACTELION PHARMACEUTICALS LTD. (CH) 2007-05-31 US claimed
EP-4671252-A4 HETEROCYCLIC-SUBSTITUTED PYRIMIDOPYRAN COMPOUND AND USE THEREOF D3 BIO WUXI CO LTD (CN) 2026-05-27 EP disclosed
CN-116761799-B Pyrimidopyran compounds 德昇济医药(无锡)有限公司 2026-03-06 CN disclosed
CN-116761799-B Pyrimidopyran compounds 德昇济医药(无锡)有限公司 2026-03-06 CN disclosed
WO-2026046397-A1 HETEROCYCLIC SUBSTITUTED PYRIMIDOPYRAN COMPOUNDS AND USES THEREOF D3 BIO (WUXI) CO., LTD. (CN) 2026-03-05 WO disclosed
WO-2026046397-A1 HETEROCYCLIC SUBSTITUTED PYRIMIDOPYRAN COMPOUNDS AND USES THEREOF D3 BIO (WUXI) CO., LTD. (CN) 2026-03-05 WO disclosed
EP-4671252-A1 HETEROCYCLIC-SUBSTITUTED PYRIMIDOPYRAN COMPOUND AND USE THEREOF D3 Bio(Wuxi) Co., Ltd. (CN) 2025-12-31 EP disclosed
WO-2025195335-A1 HETEROCYCLIC SUBSTITUTED PYRIMIDOPYRAN COMPOUNDS AND THEIR APPLICATIONS D3 BIO (WUXI) CO., LTD. (CN) 2025-09-25 WO disclosed
WO-2025195335-A1 HETEROCYCLIC SUBSTITUTED PYRIMIDOPYRAN COMPOUNDS AND THEIR APPLICATIONS D3 BIO (WUXI) CO., LTD. (CN) 2025-09-25 WO disclosed
WO-2009047514-A1 [1,2,4]TRIAZOLO[1,5-A]PYRIDINE AND [1,2,4]TRIAZOLO[1,5-C]PYRIMIDINE COMPOUNDS AND THEIR USE CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2009-04-16 WO disclosed
EP-1663993-B1 GUANIDINE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2008-03-12 EP disclosed
US-20070123510-A1 Guanidine derivatives ACTELION PHARMACEUTICALS LTD. (CH) 2007-05-31 US disclosed
US-6448256-B1 PRECURSORS OF N-SUBSTITUTED DERIVATIVES OF 6-AMINOURACILS, 6-AMINOISOCYTOSINES, GUANINES AND 2-AMINOADENINES HAVING A CLEAVABLE ESTER GROUP; GREATER WATER SOLUBILITY AND ORAL BIOAVAILABILITY; TREATING GRAM POSITIVE BACTERIAL INFECTIONS UNIVERSITY OF MASSACHUSETTS 2002-09-10 US disclosed
EP-1185517-A1 ANTIBIOTIC PRODRUGS University of Massachusetts (US) 2002-03-13 EP disclosed
WO-2000071523-A1 ANTIBIOTIC PRODRUGS UNIVERSITY OF MASSACHUSETTS (US) 2000-11-30 WO disclosed
EP-1022278-A1 TETRACYCLICAL DERIVATIVES FROM PYRIMIDINE Ashkinazi, Rimma Iliinichna (RU) 2000-07-26 EP disclosed
US-6071905-A TREATING TUBERCULOSIS, MYCOBACTERIOSIS, VIRAL AND IMMUNE DISEASES, CHLAMYDIA INFECTIONS, ANTITUMOR AND -CARCINOGENIC AGENTS; MICROBIOCIDES, IN PARTICULAR TO MYCOBACTERIA RESISTANT TO ISONIAZIDE; STIMULANTES INTERFERONS NATURAL DRUG SCIENCES, LLC (US) 2000-06-06 US disclosed
EP-0276057-A2 Piperazinylpyrimidines as beta-adrenergic receptor blocking agents MERCK & CO. INC. (US) 1988-07-27 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070123510-A1 Guanidine derivatives NPFFR1, NPFFR2, OGFR CA1 4362/4885CA9 4717/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.