SCHEMBL21848083

SCHEMBL21848083

CC(C)(C)C1[C@@H](C(N)c2ccccc2)CCN1C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45
TSHR P16473 1/20 0.45
MAPK1 P28482 1/20 0.45
HSD17B10 Q99714 1/20 0.45
RIPK1 Q13546 3/20 0.40
DPP4 P27487 5/20 0.38
AGTR2 P50052 4/20 0.36
OPRM1 P35372 2/20 0.36
OPRD1 P41143 2/20 0.36
OPRK1 P41145 2/20 0.36
OPRL1 P41146 2/20 0.36
KDM4E B2RXH2 1/20 0.36
DPP7 Q9UHL4 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
DPP8 Q6V1X1 1/20 0.35
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22077636 1.00 CYP3A4 (0.45) CYP3A4CYP1A2CYP2D6TSHRMAPK1
SCHEMBL3807599 0.77 RIPK1 (0.43) CYP2D6RIPK1DPP4KDM4EDPP8
SCHEMBL22436253 0.77 TDP1 (0.33) RIPK1OPRM1
SCHEMBL25411430 0.76 CYP2D6 (0.32) CYP2D6RIPK1DPP4LMNA
SCHEMBL859746 0.73 RIPK1 (0.35) CYP3A4RIPK1KDM4EMEN1KMT2A
SCHEMBL23826433 0.71 DPP4 (0.34) DPP4DPP7DPP8
SCHEMBL23825766 0.71 DPP4 (0.34) DPP4DPP7DPP8
SCHEMBL23826651 0.70 DPP4 (0.33) DPP4DPP7DPP8
SCHEMBL3533635 0.70 DPP4 (0.51) CYP3A4CYP1A2CYP2D6TSHRMAPK1
SCHEMBL3533638 0.70 DPP4 (0.51) CYP3A4CYP1A2CYP2D6TSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3640242-A1 ROCK-INHIBITING COMPOUND AND USES THEREOF Hitgen Ltd. (CN) 2020-04-22 EP disclosed