SCHEMBL21856901

SCHEMBL21856901

O=S(=O)(Nc1cccc(-c2nn[nH]n2)c1)c1ccc(-c2ccon2)s1

nearest known ligand 0.76

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PFKFB3 Q16875 13/20 0.76
PFKFB4 Q16877 8/20 0.71
LNPEP Q9UIQ6 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21857152 0.87 PFKFB3 (1.00) PFKFB3PFKFB4
SCHEMBL21857715 0.84 PFKFB3 (0.73) PFKFB3PFKFB4
SCHEMBL21857876 0.84 PFKFB3 (0.82) PFKFB3PFKFB4LNPEP
SCHEMBL21857049 0.84 PFKFB3 (0.86) PFKFB3PFKFB4LNPEP
SCHEMBL21857540 0.83 PFKFB3 (0.84) PFKFB3PFKFB4LNPEP
SCHEMBL21857117 0.83 PFKFB3 (1.00) PFKFB3PFKFB4
SCHEMBL21857632 0.82 PFKFB3 (1.00) PFKFB3PFKFB4
SCHEMBL794168 0.82 PFKFB3 (0.60) PFKFB3PFKFB4
SCHEMBL21857895 0.82 PFKFB4 (0.84) PFKFB3PFKFB4LNPEP
SCHEMBL21857534 0.82 PFKFB3 (1.00) PFKFB3PFKFB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113396145-A PFKFB3 inhibitors and uses thereof 盖罗发现有限责任公司 2021-09-14 CN disclosed
WO-2020080979-A1 PFKFB3 INHIBITORS AND THEIR USES GERO DISCOVERY LIMITED LIABILITY COMPANY (RU) 2020-04-23 WO disclosed