SCHEMBL21858034

SCHEMBL21858034

C(#Cc1cccc2ccccc12)c1cccc2[c]cccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHAT P28329 1/20 0.50
GRM5 P41594 1/20 0.43
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
ALDH1A1 P00352 6/20 0.38
CYP2A6 P11509 3/20 0.38
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
MITF O75030 1/20 0.36
MAPT P10636 1/20 0.36
HTT P42858 1/20 0.36
RAD52 P43351 1/20 0.36
HRH3 Q9Y5N1 4/20 0.35
ACACB O00763 1/20 0.35
HSD17B10 Q99714 4/20 0.34
TSHR P16473 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
KDM4E B2RXH2 1/20 0.34
POLB P06746 1/20 0.34
CYP1A2 P05177 4/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21858021 0.93 CHAT (0.46) CHATGRM5CA1CA2ALDH1A1
SCHEMBL21858099 0.84 CHAT (0.49) CHATGRM5CA1CA2ALDH1A1
SCHEMBL21858110 0.84 CHAT (0.45) CHATGRM5CA2ALDH1A1MEN1
SCHEMBL21858085 0.82 CHAT (0.49) CHATGRM5CA1CA2ALDH1A1
SCHEMBL21858027 0.82 CHAT (0.49) CHATGRM5CA1CA2ALDH1A1
SCHEMBL21858058 0.82 CHAT (0.42) CHATGRM5CA1CA2HRH3
SCHEMBL2776015 0.82 CHAT (0.60) CHATGRM5CA1CA2ALDH1A1
SCHEMBL29661843 0.82 CHAT (0.60) CHATGRM5CA1CA2ALDH1A1
SCHEMBL21858053 0.80 CHAT (0.49) CHATGRM5CA1CA2ALDH1A1
SCHEMBL6364668 0.80 CHAT (0.58) CHATGRM5CA1CA2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112955422-B polycyclic compound 三菱瓦斯化学株式会社 2023-08-22 CN claimed
US-20210355058-A1 POLYCYCLIC COMPOUNDS MITSUBISHI GAS CHEMICAL CO (JP) 2021-11-18 US claimed
US-20210340317-A1 POLYCYCLIC COMPOUNDS REUTER CHEMISCHE APPARATEBAU E.K. (DE) 2021-11-04 US claimed
CN-112955422-A Polycyclic compounds 三菱瓦斯化学株式会社 2021-06-11 CN claimed
WO-2020080558-A1 POLYCYCLIC COMPOUNDS MITSUBISHI GAS CHEMICAL COMPANY, INC. (JP) 2020-04-23 WO claimed
WO-2020079225-A1 POLYCYCLIC COMPOUNDS REUTER CHEMISCHE APPARATEBAU E.K. (DE) 2020-04-23 WO claimed
CN-112955422-B polycyclic compound 三菱瓦斯化学株式会社 2023-08-22 CN disclosed
US-20210355058-A1 POLYCYCLIC COMPOUNDS MITSUBISHI GAS CHEMICAL CO (JP) 2021-11-18 US disclosed
US-20210340317-A1 POLYCYCLIC COMPOUNDS REUTER CHEMISCHE APPARATEBAU E.K. (DE) 2021-11-04 US disclosed
CN-112955422-A Polycyclic compounds 三菱瓦斯化学株式会社 2021-06-11 CN disclosed
WO-2020080558-A1 POLYCYCLIC COMPOUNDS MITSUBISHI GAS CHEMICAL COMPANY, INC. (JP) 2020-04-23 WO disclosed
WO-2020079225-A1 POLYCYCLIC COMPOUNDS REUTER CHEMISCHE APPARATEBAU E.K. (DE) 2020-04-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210340317-A1 POLYCYCLIC COMPOUNDS CBR1, C1R, CBR3 CHAT 3261/4885GRM5 2617/4885CA1 2606/4885
US-20210355058-A1 POLYCYCLIC COMPOUNDS CBR1, CBR3, C1R CHAT 3179/4885GRM5 2703/4885CA1 2553/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.