SCHEMBL2185958

SCHEMBL2185958

O=C(Cn1nccn1)N(C(=O)C1CC(Cc2ccccc2Cl)CN1)c1ccc(Oc2ccc(F)cc2)cc1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.37
S1PR1 P21453 2/20 0.37
MLNR O43193 3/20 0.32
SCN9A Q15858 3/20 0.32
TP53 P04637 2/20 0.31
MAPK8 P45983 1/20 0.31
NPBWR1 P48145 1/20 0.31
TACR1 P25103 2/20 0.31
MAPT P10636 1/20 0.31
HRH3 Q9Y5N1 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP3A4 P08684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2210631 0.92 CYP2C9 (0.38) CYP2C9S1PR1SCN9AHRH3CYP2D6
SCHEMBL2169856 0.87 CYP2C9 (0.45) CYP2C9S1PR1MLNRHRH3CYP2D6
SCHEMBL3122969 0.86 CYP2C9 (0.40) CYP2C9S1PR1HRH3CYP2D6
SCHEMBL2172041 0.86 CYP2C9 (0.40) CYP2C9S1PR1HRH3CYP2D6
SCHEMBL2170954 0.77 S1PR1 (0.41) CYP2C9S1PR1CYP2D6CYP3A4
SCHEMBL2357176 0.77 HRH3 (0.37) CYP2C9S1PR1MAPTHRH3CYP2D6
SCHEMBL2187351 0.75 S1PR1 (0.41) CYP2C9S1PR1HRH3CYP2D6CYP3A4
SCHEMBL2170534 0.75 CYP2C9 (0.48) CYP2C9S1PR1MLNRHRH3CYP2D6
SCHEMBL3258058 0.75 CYP2D6 (0.41) CYP2C9S1PR1HRH3CYP2D6
SCHEMBL2205673 0.75 S1PR1 (0.51) CYP2C9S1PR1MLNRHRH3CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346821-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS Exelixis, Inc. (US) 2011-07-27 EP disclosed