SCHEMBL2172041

SCHEMBL2172041

O=C(Cn1nccn1)N(C(=O)[C@@H]1C[C@@H](Cc2cccc(Cl)c2)CN1)c1ccc(Oc2ccc(F)cc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.40
S1PR1 P21453 2/20 0.40
F2 P00734 3/20 0.36
HRH3 Q9Y5N1 2/20 0.36
FAAH O00519 3/20 0.34
MMP13 P45452 1/20 0.33
CYP2D6 P10635 1/20 0.32
ALOX5 P09917 1/20 0.32
OPRM1 P35372 1/20 0.32
SIGMAR1 Q99720 1/20 0.31
CACNA1G O43497 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3122969 1.00 CYP2C9 (0.40) CYP2C9S1PR1F2HRH3FAAH
SCHEMBL2169856 0.91 CYP2C9 (0.45) CYP2C9S1PR1F2HRH3MMP13
SCHEMBL2185958 0.86 CYP2C9 (0.37) CYP2C9S1PR1HRH3CYP2D6
SCHEMBL2210631 0.84 CYP2C9 (0.38) CYP2C9S1PR1HRH3CYP2D6OPRM1
SCHEMBL2357176 0.79 HRH3 (0.37) CYP2C9S1PR1F2HRH3MMP13
SCHEMBL2170534 0.79 CYP2C9 (0.48) CYP2C9S1PR1F2HRH3MMP13
SCHEMBL2184284 0.78 CYP2C9 (0.47) CYP2C9S1PR1HRH3CYP2D6OPRM1
SCHEMBL2352992 0.77 MEN1 (0.37) CYP2C9S1PR1F2HRH3CYP2D6
SCHEMBL2205673 0.77 S1PR1 (0.51) CYP2C9S1PR1F2HRH3MMP13
SCHEMBL2350633 0.76 OPRM1 (0.39) CYP2C9S1PR1HRH3CYP2D6OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346821-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS Exelixis, Inc. (US) 2011-07-27 EP disclosed