SCHEMBL21863291

SCHEMBL21863291

CCc1cn(-c2cccc(OC(F)(F)F)c2)nn1

nearest known ligand 0.73

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
RXRA P19793 15/20 0.73
GRIN1 Q05586 15/20 0.73
GRIN2B Q13224 15/20 0.73
KCNH2 Q12809 4/20 0.70
NOTUM Q6P988 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19211503 0.86 RXRA (0.68) RXRAGRIN1GRIN2BKCNH2NOTUM
SCHEMBL27430549 0.86 RXRA (0.68) RXRAGRIN1GRIN2BKCNH2NOTUM
SCHEMBL19219461 0.85 RXRA (1.00) RXRAGRIN1GRIN2B
SCHEMBL17502335 0.83 KCNH2 (1.00) RXRAGRIN1GRIN2BKCNH2
SCHEMBL23346078 0.83 NOTUM (0.60) RXRAGRIN1GRIN2BNOTUM
SCHEMBL17502221 0.82 KCNH2 (1.00) RXRAGRIN1GRIN2BKCNH2
SCHEMBL19219445 0.81 RXRA (1.00) RXRAGRIN1GRIN2B
SCHEMBL19219447 0.80 RXRA (1.00) RXRAGRIN1GRIN2B
SCHEMBL19219460 0.79 RXRA (1.00) RXRAGRIN1GRIN2B
SCHEMBL19219454 0.78 RXRA (1.00) RXRAGRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3180329-B1 TRIAZOLES AS NR2B RECEPTOR INHIBITORS JANSSEN PHARMACEUTICALS INC (US) 2020-03-18 EP disclosed