SCHEMBL21865764

SCHEMBL21865764

Cc1cc(OC(F)(F)F)cc2c1NCC2C

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 3/20 0.33
PTGS2 P35354 3/20 0.33
AR P10275 1/20 0.32
HTR2A P28223 5/20 0.31
HTR2C P28335 5/20 0.31
HTR2B P41595 5/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31607544 0.74 HTR2C (0.40) ARHTR2AHTR2CHTR2B
SCHEMBL5675008 0.70 HTR2C (0.40) HTR2AHTR2CHTR2B
SCHEMBL15189277 0.66 FFAR4 (0.42) PTGS1PTGS2
SCHEMBL21866083 0.65 AR (0.38) ARHTR2AHTR2CHTR2B
SCHEMBL16707469 0.65 PTGS1 (0.39) PTGS1PTGS2
SCHEMBL23273109 0.63 PTGS1 (0.38) PTGS1PTGS2
SCHEMBL21603434 0.63 TP53 (0.44) PTGS1PTGS2
SCHEMBL31607527 0.63 MEN1 (0.58) HTR2AHTR2CHTR2B
SCHEMBL19422711 0.62 HSPA9 (0.33) PTGS1PTGS2HTR2AHTR2CHTR2B
SCHEMBL16954442 0.61 TRPV1 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3636643-A1 NUCLEAR RECEPTOR MODULATORS (ROR) FOR THE TREATMENT OF INFLAMMATORY AND AUTOIMMUNE DISEASES AbbVie Inc. (US) 2020-04-15 EP disclosed