SCHEMBL21869760

SCHEMBL21869760

COc1ccc(COC(=O)[C@@H]2CCC(=O)N2Cc2ccc(C)cc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.60
GAA P10253 2/20 0.49
POLB P06746 1/20 0.48
ALDH1A1 P00352 2/20 0.48
KDM4E B2RXH2 1/20 0.48
MAPT P10636 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.46
HCRTR1 O43613 2/20 0.46
HCRTR2 O43614 2/20 0.46
HDAC1 Q13547 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21869762 1.00 KMT2A (0.60) KMT2AGAAPOLBALDH1A1KDM4E
SCHEMBL21869749 0.95 KMT2A (0.52) KMT2AHCRTR1HCRTR2HDAC1HDAC6
SCHEMBL21869750 0.93 KMT2A (0.67) KMT2AGAAALDH1A1KDM4EMAPT
SCHEMBL21869759 0.92 KMT2A (0.49) KMT2AHCRTR1HCRTR2HDAC1HDAC6
SCHEMBL21869748 0.91 HDAC1 (0.53) KMT2AHCRTR1HCRTR2HDAC1HDAC6
SCHEMBL28669317 0.91 HDAC1 (0.53) KMT2AHCRTR1HCRTR2HDAC1HDAC6
SCHEMBL21869826 0.91 HDAC1 (0.53) KMT2AHCRTR1HCRTR2HDAC1HDAC6
SCHEMBL21869752 0.90 KMT2A (0.47) KMT2AHCRTR1HCRTR2HDAC1HDAC6
SCHEMBL21869800 0.90 HCRTR2 (0.52) KMT2AGAAPOLBALDH1A1CYP2C19
SCHEMBL21869753 0.90 KMT2A (0.63) KMT2AGAAALDH1A1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109180552-B Substituted 5-oxo pyrrolidine derivative and preparation method and application thereof 沈阳药科大学 2021-10-26 CN disclosed
WO-2020063388-A1 SUBSTITUTED 5-OXOPYRROLIDINE DERIVATIVE, PREPARATION METHOD THEREFOR AND USE THEREOF 沈阳药科大学 2020-04-02 WO disclosed