SCHEMBL21869752

SCHEMBL21869752

COc1ccc(CN2C(=O)CC[C@H]2C(=O)OCc2ccc(N)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.47
HCRTR1 O43613 2/20 0.45
HCRTR2 O43614 2/20 0.45
HDAC1 Q13547 6/20 0.43
HDAC6 Q9UBN7 1/20 0.43
HDAC2 Q92769 4/20 0.43
HDAC3 O15379 2/20 0.43
FABP7 O15540 1/20 0.43
FABP5 Q01469 1/20 0.43
CYP19A1 P11511 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21869749 0.94 KMT2A (0.52) KMT2AHCRTR1HCRTR2HDAC1HDAC6
SCHEMBL21869759 0.91 KMT2A (0.49) KMT2AHCRTR1HCRTR2HDAC1HDAC6
SCHEMBL28669317 0.90 HDAC1 (0.53) KMT2AHCRTR1HCRTR2HDAC1HDAC6
SCHEMBL21869748 0.90 HDAC1 (0.53) KMT2AHCRTR1HCRTR2HDAC1HDAC6
SCHEMBL21869826 0.90 HDAC1 (0.53) KMT2AHCRTR1HCRTR2HDAC1HDAC6
SCHEMBL21869760 0.90 KMT2A (0.60) KMT2AHCRTR1HCRTR2HDAC1HDAC6
SCHEMBL21869762 0.90 KMT2A (0.60) KMT2AHCRTR1HCRTR2HDAC1HDAC6
SCHEMBL21869800 0.89 HCRTR2 (0.52) KMT2AHCRTR1HCRTR2HDAC1HDAC2
SCHEMBL21869751 0.89 KMT2A (0.61) KMT2AHDAC1HDAC6
SCHEMBL21869794 0.87 HDAC1 (0.50) KMT2AHDAC1HDAC6HDAC2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109180552-B Substituted 5-oxo pyrrolidine derivative and preparation method and application thereof 沈阳药科大学 2021-10-26 CN disclosed
WO-2020063388-A1 SUBSTITUTED 5-OXOPYRROLIDINE DERIVATIVE, PREPARATION METHOD THEREFOR AND USE THEREOF 沈阳药科大学 2020-04-02 WO disclosed