SCHEMBL21884022

SCHEMBL21884022

N#Cc1c(-n2c3ccccc3c3ccccc32)c(-n2c3ccccc3c3ccccc32)c(-n2c3ccccc3c3ccccc32)c(-n2c3ccccc3c3cc(-c4ccc5c(c4)c4ccccc4n5-c4cccc(-c5cccc(-n6c7ccccc7c7ccccc76)c5)c4)ccc32)c1-n1c2ccccc2c2ccccc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.40
ATM Q13315 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ALDH1A1 P00352 5/20 0.34
HPGD P15428 3/20 0.34
LMNA P02545 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MAPT P10636 1/20 0.33
CASP1 P29466 1/20 0.33
HSD17B10 Q99714 1/20 0.33
TSPO P30536 1/20 0.33
CYP11B2 P19099 1/20 0.33
PTGER4 P35408 2/20 0.32
EGFR P00533 1/20 0.32
SRC P12931 1/20 0.32
PDE9A O76083 1/20 0.32
PDE1C Q14123 1/20 0.32
MAPK1 P28482 1/20 0.32
STAT3 P40763 1/20 0.32
FAAH O00519 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23979238 1.00 KDM4E (0.40) KDM4EATML3MBTL1ALDH1A1HPGD
SCHEMBL17570302 0.90 KDM4E (0.40) KDM4EATML3MBTL1ALDH1A1HPGD
SCHEMBL21377993 0.89 KDM4E (0.42) KDM4EATML3MBTL1ALDH1A1HPGD
SCHEMBL21884031 0.89 TSPO (0.40) KDM4EATML3MBTL1ALDH1A1HPGD
SCHEMBL23979224 0.89 TSPO (0.40) KDM4EATML3MBTL1ALDH1A1HPGD
SCHEMBL21765765 0.89 TSPO (0.40) KDM4EATML3MBTL1ALDH1A1HPGD
SCHEMBL21840849 0.89 TSPO (0.40) KDM4EATML3MBTL1ALDH1A1HPGD
SCHEMBL23263992 0.89 TSPO (0.40) KDM4EATML3MBTL1ALDH1A1HPGD
SCHEMBL21840840 0.89 TSPO (0.40) KDM4EATML3MBTL1ALDH1A1HPGD
SCHEMBL21884024 0.89 TSPO (0.40) KDM4EATML3MBTL1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020059326-A1 BENZONITRILE DERIVATIVE AND MANUFACTURING METHOD THEREFOR, INK COMPOSITION, ORGANIC ELECTROLUMINESCENT ELEMENT MATERIAL, LIGHT-EMITTING MATERIAL, CHARGE TRANSPORT MATERIAL, LIGHT-EMITTING THIN FILM, AND ORGANIC ELECTROLUMINESCENT ELEMENT コニカミノルタ株式会社 2020-03-26 WO disclosed
WO-2020059520-A1 BENZONITRILE DERIVATIVE AND MANUFACTURING METHOD THEREFOR, INK COMPOSITION, ORGANIC ELECTROLUMINESCENT ELEMENT MATERIAL, LIGHT-EMITTING MATERIAL, CHARGE TRANSPORT MATERIAL, LIGHT-EMITTING THIN FILM, AND ORGANIC ELECTROLUMINESCENT ELEMENT コニカミノルタ株式会社 2020-03-26 WO disclosed