SCHEMBL2189355

SCHEMBL2189355

CC(C)c1ccc(NC(=O)NCc2nc(C(=O)NCCc3cccc(Cl)c3)cs2)cc1.CC(C)c1ccc(NC(=O)NCc2nc(C(=O)NCCc3ccccc3F)cs2)cc1.CCOc1cccc(CCNC(=O)c2csc(CNC(=O)COc3ccc(OC(F)(F)F)cc3)n2)c1.C[C@H](CNC(=O)c1csc(CNC(=O)COc2ccc(OC(F)(F)F)cc2)n1)c1ccccc1.O=C(COc1ccc(OC(F)(F)F)cc1)NCc1nc(C(=O)NCCc2ccc(F)cc2)cs1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.37
MAPT P10636 2/20 0.35
TP53 P04637 1/20 0.35
RAF1 P04049 1/20 0.35
TRPV1 Q8NER1 1/20 0.35
ALDH1A1 P00352 2/20 0.35
SLC2A1 P11166 1/20 0.35
RORC P51449 3/20 0.34
SGMS1 Q86VZ5 2/20 0.33
GAA P10253 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
IGF1R P08069 2/20 0.33
HTRA1 Q92743 1/20 0.33
EPHX1 P07099 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
KMT2A Q03164 1/20 0.32
LMNA P02545 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2189359 0.89 CNR1 (0.33) CNR1MAPTTP53RAF1TRPV1
SCHEMBL4387708 0.78 TRPV1 (0.44) CNR1MAPTTP53RAF1TRPV1
SCHEMBL283213 0.77 TRPV1 (0.58) CNR1MAPTTP53TRPV1SGMS1
SCHEMBL2171624 0.76 CNR1 (0.51) CNR1MAPTTP53ALDH1A1GAA
SCHEMBL2174484 0.76 IGF1R (0.49) MAPTTP53TRPV1SLC2A1GAA
SCHEMBL2186611 0.75 TRPV1 (0.48) MAPTTP53TRPV1SGMS1IGF1R
SCHEMBL4392406 0.75 ALDH1A1 (0.43) MAPTALDH1A1GAAKMT2ASMN1; SMN2
SCHEMBL5668846 0.75 IGF1R (0.47) MAPTGAAIGF1RRAB9AKMT2A
SCHEMBL4383724 0.75 ALDH1A1 (0.43) MAPTALDH1A1GAAKMT2ASMN1; SMN2
SCHEMBL4395355 0.75 ALDH1A1 (0.43) MAPTALDH1A1GAAKMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7973061-B2 Anaplastic lymphoma kinase modulators and methods of use EXELIXIS, INC. (US) 2011-07-05 US claimed