SCHEMBL21899343

SCHEMBL21899343

COCc1cncc(Cl)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 3/20 0.41
S1PR4 O95977 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
ALDH1A1 P00352 3/20 0.33
MAPT P10636 2/20 0.33
MRGPRX4 Q96LA9 1/20 0.33
NOTUM Q6P988 1/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
PKM P14618 1/20 0.33
LMNA P02545 2/20 0.32
TDP1 Q9NUW8 2/20 0.32
TUBB4A P04350 1/20 0.32
TUBB P07437 1/20 0.32
TUBA3C P0DPH7 1/20 0.32
TUBA1B P68363 1/20 0.32
TUBA4A P68366 1/20 0.32
TUBB4B P68371 1/20 0.32
TUBB3 Q13509 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4264181 0.84 LMNA (0.38) S1PR4ALDH1A1MAPTMRGPRX4CYP11B1
SCHEMBL32666839 0.82 CDK2 (0.38) CDK2HDAC1HDAC6
SCHEMBL8190613 0.77
SCHEMBL13700992 0.76 LMNA (0.37) ALDH1A1MAPTCYP11B1CYP11B2PKM
SCHEMBL30539179 0.75 HDAC1 (0.36) CDK2HDAC1HDAC6
SCHEMBL25783036 0.75 HDAC1 (0.36) CDK2HDAC1HDAC6
SCHEMBL20772527 0.75 CDK2 (0.35) CDK2HTR2A
SCHEMBL22772487 0.75
SCHEMBL22576285 0.74 CDK2 (0.41) CDK2ALDH1A1MAPTLMNAKDM4E
SCHEMBL28105653 0.74 CDK2 (0.38) CDK2HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020081999-A1 ANDROGEN RECEPTOR MODULATORS AND METHODS FOR THEIR USE ESSA PHARMA, INC. (CA) 2020-04-23 WO disclosed