SCHEMBL21920109

SCHEMBL21920109

CCCC[C@@H](CCC)Nc1nc(NC(C)=O)ncc1OCc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 7/20 0.44
PPIA P62937 1/20 0.41
PTGES O14684 1/20 0.40
ALOX5 P09917 1/20 0.40
KCNH2 Q12809 1/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
ADORA1 P30542 1/20 0.39
TLR7 Q9NYK1 2/20 0.38
TLR8 Q9NR97 3/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
APP P05067 1/20 0.38
ACHE P22303 1/20 0.38
CYP19A1 P11511 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13195028 0.94 KCNH2 (0.47) BRD4PPIAPTGESALOX5KCNH2
SCHEMBL15469718 0.93 TLR8 (0.46) BRD4PPIAPTGESALOX5KCNH2
SCHEMBL15469765 0.92 KCNH2 (0.45) BRD4PPIAKCNH2CYP11B1CYP11B2
SCHEMBL15469717 0.87 BRD4 (0.42) BRD4PPIAPTGESALOX5CYP11B1
SCHEMBL17123640 0.86 TLR8 (0.42) BRD4KCNH2TLR7TLR8
SCHEMBL20386619 0.83 KCNH2 (0.48) KCNH2TLR7TLR8CYP1A2CYP2D6
SCHEMBL17123643 0.83 CYP1A2 (0.52) BRD4PPIACYP11B1CYP11B2ADORA3
SCHEMBL20386594 0.81 CYP1A2 (0.48) BRD4PPIACYP11B1CYP11B2ADORA3
SCHEMBL15470054 0.79 KCNH2 (0.59) KCNH2TLR7TLR8CYP1A2CYP2D6
SCHEMBL19274231 0.79 KCNH2 (0.53) KCNH2TLR7TLR8CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2903967-B3 ACYLAMINOPYRIMIDINE DERIVATIVES FOR THE TREATMENT OF VIRAL INFECTIONS AND FURTHER DISEASES JANSSEN SCIENCES IRELAND UNLIMITED CO (IE) 2020-04-15 EP disclosed