SCHEMBL21921098

SCHEMBL21921098

CCC(F)(F)COc1ccc(C)nc1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 4/20 0.39
CHRNA4 P43681 4/20 0.39
KMT2A Q03164 2/20 0.39
CHRNB1 P11230 1/20 0.39
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
CHRNB3 Q05901 1/20 0.39
GRM5 P41594 1/20 0.39
MAPT P10636 1/20 0.39
ADRB2 P07550 1/20 0.35
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20231023 0.85 CHRNB2 (0.38) CHRNB2CHRNA4KMT2ACHRNB1CHRNB4
SCHEMBL506299 0.84 CHRNB2 (0.42) CHRNB2CHRNA4KMT2ACHRNB1CHRNB4
SCHEMBL20233868 0.83 CHRNB2 (0.35) CHRNB2CHRNA4KMT2ACHRNB1CHRNB4
SCHEMBL21182267 0.81 CHRNB2 (0.40) CHRNB2CHRNA4KMT2ACHRNB1CHRNB4
SCHEMBL26401540 0.79 CHRNB2 (0.39) CHRNB2CHRNA4KMT2ACHRNB1CHRNB4
SCHEMBL13020439 0.78 CHRNB2 (0.45) CHRNB2CHRNA4KMT2ACHRNB1CHRNB4
SCHEMBL26401405 0.78 HTT (0.43) CHRNB2CHRNA4KMT2ACHRNB1CHRNB4
SCHEMBL26401534 0.77 CHRNB2 (0.40) CHRNB2CHRNA4CHRNB1CHRNB4CHRNA3
SCHEMBL20441137 0.76 KMT2A (0.40) CHRNB2CHRNA4KMT2ACHRNB1CHRNB4
SCHEMBL2669046 0.75 NQO1 (0.56) CHRNB2CHRNA4KMT2ACHRNB1CHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3632899-A1 ARYL SUBSTITUTED CARBOXAMIDE DERIVATIVES AS CALCIUM OR SODIUM CHANNEL BLOCKERS RaQualia Pharma Inc. (JP) 2020-04-08 EP disclosed