SCHEMBL21923085

SCHEMBL21923085

O=C(Nc1cccc(F)c1)C1CCOC1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIP5K1C O60331 3/20 0.54
PIK3CA P42336 3/20 0.54
MAP4K4 O95819 1/20 0.54
MAPK10 P53779 3/20 0.52
MAPK8 P45983 2/20 0.52
MAPK14 Q16539 2/20 0.52
ACKR3 P25106 1/20 0.52
ALDH1A1 P00352 1/20 0.51
POLB P06746 1/20 0.51
HTT P42858 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
MGLL Q99685 1/20 0.51
PIP5K1B O14986 1/20 0.51
PIP5K1A Q99755 1/20 0.51
HSD17B10 Q99714 1/20 0.50
MAPT P10636 1/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
MEN1 O00255 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28872344 0.92 SMN1; SMN2 (0.56) PIP5K1CPIK3CAMAP4K4MAPK10MAPK8
SCHEMBL27923186 0.84 GAA (0.62) ALDH1A1POLBHTTTDP1SMN1; SMN2
SCHEMBL8278939 0.83 NPSR1 (0.68) PIP5K1CPIK3CAMAP4K4MAPK10MAPK8
SCHEMBL29076764 0.81 NPSR1 (0.63) ALDH1A1POLBHTTTDP1SMN1; SMN2
SCHEMBL17896347 0.80 ACKR3 (0.57) PIP5K1CPIK3CAMAP4K4MAPK10MAPK8
SCHEMBL16401329 0.80 ALDH1A1 (0.67) ALDH1A1SMN1; SMN2MGLLNPC1RAB9A
SCHEMBL27347877 0.78 F10 (0.63) ALDH1A1POLBHTTTDP1SMN1; SMN2
SCHEMBL31401961 0.77 KMT2A (0.56) PIP5K1CPIK3CAMAP4K4MAPK10MAPK8
Hydrochloric Acid SCHEMBL30690907 0.77 F10 (0.61) ALDH1A1POLBHTTTDP1SMN1; SMN2
Hydrochloric Acid SCHEMBL27146052 0.77 F10 (0.61) ALDH1A1POLBHTTTDP1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2855459-B1 AMINOQUINAZOLINE AND PYRIDOPYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2020-04-29 EP disclosed