SCHEMBL21940787

SCHEMBL21940787

Cc1cc(C#N)nnc1N1CC(F)(F)C1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 1/20 0.35
ALDH1A1 P00352 3/20 0.35
HPGD P15428 3/20 0.35
KDM4E B2RXH2 2/20 0.35
HSD17B10 Q99714 2/20 0.35
RECQL P46063 1/20 0.35
LRRK2 Q5S007 1/20 0.34
P4HTM Q9NXG6 2/20 0.34
TSHR P16473 1/20 0.33
KHK P50053 1/20 0.33
MBOAT4 Q96T53 1/20 0.32
AKT1 P31749 1/20 0.31
AKT2 P31751 1/20 0.31
AKT3 Q9Y243 1/20 0.31
NOS3 P29474 1/20 0.30
NOS1 P29475 1/20 0.30
NOS2 P35228 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20606768 0.88 LRRK2 (0.40) ALDH1A1HPGDKDM4EHSD17B10RECQL
SCHEMBL21941079 0.77 LRRK2 (0.38) ALDH1A1HPGDKDM4EHSD17B10RECQL
SCHEMBL21940582 0.73 KDM4E (0.44) ALDH1A1HPGDKDM4EHSD17B10TSHR
SCHEMBL21940293 0.73 KDM4E (0.44) ALDH1A1HPGDKDM4EHSD17B10TSHR
SCHEMBL21940800 0.73 KDM4E (0.44) ALDH1A1HPGDKDM4EHSD17B10TSHR
SCHEMBL21940802 0.73 KDM4E (0.44) ALDH1A1HPGDKDM4EHSD17B10TSHR
SCHEMBL21940505 0.72 CHRM4 (0.35) CHRM4MBOAT4NOS3NOS1NOS2
SCHEMBL21940483 0.72 P4HTM (0.36) P4HTM
SCHEMBL25148366 0.66 GRIN2D (0.32) ALDH1A1HPGDKDM4EHSD17B10RECQL
SCHEMBL25148409 0.66 PDE10A (0.39) ALDH1A1HPGDKDM4EHSD17B10RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3423445-B1 NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF FIBROSIS GALAPAGOS NV (BE) 2020-04-01 EP disclosed