SCHEMBL21941810

SCHEMBL21941810

O=C[C@@H]1CN(Cc2ccc(Oc3ccccc3)nc2)CCO1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 1/20 0.49
CNR2 P34972 2/20 0.49
RXRB P28702 1/20 0.48
DRD4 P21917 14/20 0.47
NOTUM Q6P988 1/20 0.46
SIGMAR1 Q99720 1/20 0.43
CCR5 P51681 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21902079 0.87 GRIN2B (0.64) GRIN2BCNR2DRD4
SCHEMBL21941274 0.81 GRIN2B (0.56) GRIN2BRXRBDRD4SIGMAR1
SCHEMBL21941388 0.80 RXRB (0.48) GRIN2BCNR2RXRBDRD4SIGMAR1
SCHEMBL21902097 0.79 GRIN2B (0.79) GRIN2BRXRB
SCHEMBL31663802 0.79 DRD4 (0.57) CNR2DRD4SIGMAR1
SCHEMBL1947037 0.79 DRD4 (0.57) CNR2DRD4SIGMAR1
SCHEMBL21941206 0.79 DRD4 (0.47) GRIN2BRXRBDRD4
SCHEMBL21903007 0.74 GRIN2B (0.66) GRIN2BRXRBDRD4
SCHEMBL24893024 0.71 RXRB (0.67) GRIN2BRXRBDRD4
SCHEMBL21902096 0.70 GRIN2B (0.79) GRIN2BRXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020079042-A1 4-PYRIDINYLMETHYL-MORPHOLINE DERIVATIVES AND THE USE THEREOF AS MEDICAMENT BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2020-04-23 WO disclosed