SCHEMBL2194362

SCHEMBL2194362

CC(O)Nc1cc(Nc2cccc(Br)c2)ncn1

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EGFR P00533 15/20 0.58
TNNI3K Q59H18 2/20 0.56
ERBB3 P21860 1/20 0.52
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
ABCG2 Q9UNQ0 1/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
ERBB2 P04626 1/20 0.43
TNK2 Q07912 1/20 0.43
MKNK1 Q9BUB5 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27334594 0.89 TNNI3K (0.59) EGFRTNNI3KERBB3MEN1KMT2A
SCHEMBL690653 0.77 EGFR (0.58) EGFRTNNI3KABCG2ERBB2
SCHEMBL691187 0.75 EGFR (0.57) EGFRTNNI3KABCG2ERBB2
SCHEMBL2174864 0.75 EGFR (0.71) EGFRTNNI3KERBB3
SCHEMBL691533 0.75 EGFR (0.57) EGFRTNNI3KERBB3ABCG2NPC1
SCHEMBL690552 0.74 EGFR (1.00) EGFRTNNI3KERBB3KMT2ARAB9A
SCHEMBL690934 0.73 TNNI3K (0.54) EGFRTNNI3KERBB3ABCG2ERBB2
SCHEMBL27330845 0.73 TNNI3K (0.54) EGFRTNNI3KERBB3ABCG2
SCHEMBL8798355 0.72 EGFR (0.60) EGFRTNNI3KERBB3MEN1KMT2A
SCHEMBL27322789 0.72 TNNI3K (0.63) EGFRTNNI3KERBB3ABCG2ERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079343-A2 SUBSTITUTED PYRIDINES AND PYRIMIDINES TECHNISCHE UNIVERSITAET WIEN (AT) 2011-07-07 WO disclosed