SCHEMBL8798355

SCHEMBL8798355

Cc1cccc(Nc2cc(NC(C)C)ncn2)c1

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EGFR P00533 12/20 0.60
TNNI3K Q59H18 5/20 0.58
KCNH3 Q9ULD8 1/20 0.52
POLB P06746 1/20 0.51
MEN1 O00255 1/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
KMT2A Q03164 1/20 0.47
NPSR1 Q6W5P4 1/20 0.46
HTT P42858 1/20 0.46
HIF1A Q16665 1/20 0.46
THRB P10828 1/20 0.46
ERBB3 P21860 1/20 0.45
MAPK1 P28482 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1387302 0.89 EGFR (0.72) EGFRTNNI3KMEN1NPC1RAB9A
SCHEMBL27334594 0.84 TNNI3K (0.59) EGFRTNNI3KMEN1NPC1RAB9A
SCHEMBL8798272 0.83 EGFR (0.66) EGFRTNNI3KMEN1NPC1RAB9A
SCHEMBL2782010 0.83 EGFR (0.65) EGFRTNNI3KMEN1NPC1RAB9A
SCHEMBL27318729 0.80 CFD (0.49) EGFRTNNI3KMEN1NPC1RAB9A
SCHEMBL690632 0.80 EGFR (0.62) EGFRTNNI3KMEN1NPC1RAB9A
SCHEMBL7771269 0.80 EGFR (0.66) EGFRTNNI3KPOLBMEN1NPC1
SCHEMBL8798667 0.80 EGFR (0.61) EGFRTNNI3KRAB9ANPSR1HTT
SCHEMBL7777342 0.79 EGFR (0.64) EGFRTNNI3KMEN1NPC1RAB9A
SCHEMBL2279629 0.78 EGFR (0.59) EGFRTNNI3KNPC1NPSR1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed