SCHEMBL21945819

SCHEMBL21945819

COC(=O)[C@]1(NC(=O)OC(C)(C)C)C[C@H](CC#N)C1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSK P43235 13/20 0.39
CTSS P25774 10/20 0.39
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
MAPK1 P28482 1/20 0.35
CTSL P07711 3/20 0.35
CTSB P07858 2/20 0.33
JAK2 O60674 1/20 0.32
JAK1 P23458 1/20 0.32
TYK2 P29597 1/20 0.32
JAK3 P52333 1/20 0.32
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28776848 0.88 CTSK (0.42) CTSKCTSSKMT2AMEN1MAPK1
SCHEMBL28391077 0.88 CTSK (0.42) CTSKCTSSKMT2AMEN1MAPK1
SCHEMBL21946035 0.88 CTSK (0.42) CTSKCTSSKMT2AMEN1MAPK1
SCHEMBL21946033 0.83 KMT2A (0.38) CTSKCTSSKMT2AMEN1MAPK1
SCHEMBL7926354 0.83 KMT2A (0.38) CTSKCTSSKMT2AMEN1MAPK1
SCHEMBL13763647 0.78 CTSK (0.36) CTSKCTSSKMT2AMEN1MAPK1
SCHEMBL15195550 0.78 CTSK (0.36) CTSKCTSSKMT2AMEN1MAPK1
SCHEMBL5229523 0.78 MEN1 (0.41) KMT2AMEN1MAPK1ALDH1A1
SCHEMBL5934647 0.78 MEN1 (0.41) KMT2AMEN1MAPK1ALDH1A1
SCHEMBL14416213 0.78 MEN1 (0.41) KMT2AMEN1MAPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020083336-A1 1,3,4-OXADIAZOLE-2-CYCLOBUTYL COMPOUNDS, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 南京圣和药业股份有限公司 2020-04-30 WO disclosed